SCHEMBL8226771

SCHEMBL8226771

COc1cc(C(=O)N2CCC3(CC2)CN(c2ccc(C(F)(F)F)cc2)C3c2ccc(O)cc2)cc(OC)c1OC

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.43
ALDH1A1 P00352 6/20 0.42
CYP1A2 P05177 1/20 0.42
LMNA P02545 1/20 0.42
TSHR P16473 4/20 0.42
USP2 O75604 3/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
GAA P10253 1/20 0.41
POLB P06746 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
CYP3A4 P08684 2/20 0.40
HIF1A Q16665 1/20 0.40
HRH1 P35367 1/20 0.39
ESR1 P03372 2/20 0.39
ESR2 Q92731 1/20 0.39
CYP2C9 P11712 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13596005 0.92 LMNA (0.44) PKMALDH1A1CYP1A2LMNATSHR
SCHEMBL8218870 0.89 ALDH1A1 (0.54) ALDH1A1CYP1A2LMNATSHRUSP2
SCHEMBL8228873 0.82 ALDH1A1 (0.48) PKMALDH1A1CYP1A2LMNATSHR
SCHEMBL13596002 0.81 LMNA (0.47) ALDH1A1CYP1A2LMNAL3MBTL1GAA
SCHEMBL13596003 0.81 ALDH1A1 (0.53) ALDH1A1CYP1A2LMNATSHRUSP2
SCHEMBL13596006 0.77 CACNA1H (0.50) ALDH1A1CYP1A2LMNAL3MBTL1GAA
SCHEMBL13596026 0.75 LMNA (0.48) ALDH1A1CYP1A2LMNAL3MBTL1GAA
SCHEMBL8635894 0.72 PROKR1 (0.53) PKMALDH1A1CYP1A2LMNAL3MBTL1
SCHEMBL8218775 0.71 PKM (0.48) PKMALDH1A1CYP1A2L3MBTL1GAA
SCHEMBL8202768 0.69 CACNA1H (0.52) LMNATSHRSMN1; SMN2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008033456-A1 SPIRO-CONDENSED AZETIDINE DERIVATIVES USEFUL IN TREATING PAIN, DIABETES AND DISORDERS OF LIPID METABILISM SCHERING CORPORATION (US) 2008-03-20 WO disclosed