SCHEMBL8227448

SCHEMBL8227448

CNCCCNN1C(=O)c2ccccc2C1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.43
RXRA P19793 2/20 0.40
KDM4E B2RXH2 3/20 0.40
HTR2A P28223 2/20 0.40
HRH1 P35367 2/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
RAB9A P51151 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
CHRM2 P08172 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CHRM1 P11229 1/20 0.40
DRD2 P14416 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
NFKB1 P19838 1/20 0.40
CHRM3 P20309 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30501189 0.95 SIGMAR1 (0.44) CYP1A2RXRAKDM4EHTR2AHRH1
SCHEMBL30297855 0.89 CYP1A2 (0.46) CYP1A2KDM4EALDH1A1MAPTRAB9A
SCHEMBL4950343 0.82 ASAH1 (0.56) CYP1A2ALDH1A1DRD3ASAH1
SCHEMBL31682342 0.81 GAA (0.53) CYP1A2KDM4EALDH1A1MAPTRAB9A
SCHEMBL27387263 0.81 ASAH1 (0.59) CYP1A2ALDH1A1ASAH1
SCHEMBL4079545 0.80 CYP1A2 (0.44) CYP1A2KDM4EALDH1A1MAPTRAB9A
SCHEMBL4813089 0.80 MAPT (0.45) CYP1A2KDM4EALDH1A1MAPTRAB9A
SCHEMBL13134034 0.79 CYP1A2 (0.47) CYP1A2KDM4EALDH1A1MAPTRAB9A
SCHEMBL22649169 0.79 CYP1A2 (0.43) CYP1A2KDM4EALDH1A1MAPTRAB9A
SCHEMBL28876218 0.77 CYP1A2 (0.42) CYP1A2KDM4EALDH1A1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999063933-A9 MULTIVALENT AGONISTS, PARTIAL AGONISTS AND ANTAGONISTS OF THE GABA RECEPTORS ADVANCED MEDICINE INC (US) 2000-04-27 WO disclosed