SCHEMBL8235239

SCHEMBL8235239

CN(C1CCN(C(C)(C)C)C1)S(C)(=O)=O

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.34
HTR2A P28223 8/20 0.34
HTR2C P28335 8/20 0.34
USP30 Q70CQ3 1/20 0.31
DDR1 Q08345 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26881121 1.00 PDE10A (0.34) PDE10AHTR2AHTR2CUSP30DDR1
SCHEMBL16072934 1.00 PDE10A (0.34) PDE10AHTR2AHTR2CUSP30DDR1
SCHEMBL10205104 0.89 HTR2A (0.39) HTR2AHTR2C
SCHEMBL21935713 0.86 HTR2A (0.35) PDE10AHTR2AHTR2CUSP30
SCHEMBL8260660 0.78
SCHEMBL19176922 0.77 HTR2A (0.32) HTR2AHTR2C
SCHEMBL731310 0.77 HRH4 (0.33)
SCHEMBL8260570 0.77 HRH4 (0.33)
SCHEMBL679560 0.77 HRH4 (0.33)
SCHEMBL12439352 0.76 HTR2A (0.44) HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230357242-A1 COMPOUND AS AKT KINASE INHIBITOR CHIA TAI TIANQING PHARMACEUTICAL GROUP CO., LTD. (CN) 2023-11-09 US disclosed
US-20230357242-A1 COMPOUND AS AKT KINASE INHIBITOR CHIA TAI TIANQING PHARMACEUTICAL GROUP CO., LTD. (CN) 2023-11-09 US disclosed
US-10464947-B2 Tricyclic heterocycles as BET protein inhibitors INCYTE HOLDINGS CORPORATION (US) 2019-11-05 US disclosed
US-7772239-B2 Benzoimidazolone-carboxamide compounds as 5-HT4 receptor agonists THERAVANCE, INC. (US) 2010-08-10 US disclosed
US-20080070923-A1 Benzoimidazolone-carboxamide compounds as 5-HT4 receptor agonists THERAVANCE BIOPHARMA R&D IP, LLC 2008-03-20 US disclosed
US-7317022-B2 Benzoimidazolone-carboxamide compounds as 5-HT4 receptors agonists THERAVANCE, INC. (US) 2008-01-08 US disclosed
US-20060276482-A1 Benzoimidazolone-carboxamide compounds as 5-HT4 receptors agonists THERAVANCE, INC. 2006-12-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060276482-A1 Benzoimidazolone-carboxamide compounds as 5-HT4 receptors agonists HTR4, HTR5A, HTR1A PDE10A 996/4885HTR2A 7/4885HTR2C 4/4885
US-20080070923-A1 Benzoimidazolone-carboxamide compounds as 5-HT4 receptor agonists HTR4, HTR5A, HTR1A PDE10A 979/4885HTR2A 8/4885HTR2C 4/4885
US-20230357242-A1 COMPOUND AS AKT KINASE INHIBITOR AKT2, MTOR, AKT1 PDE10A 941/4885HTR2A 3995/4885HTR2C 3480/4885
US-10464947-B2 Tricyclic heterocycles as BET protein inhibitors BRD1, BRD3, BRD2 PDE10A 4371/4885HTR2A 3190/4885HTR2C 2160/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.