SCHEMBL8237121

SCHEMBL8237121

Cc1cc(CN2CCN(C(=O)COC(c3ccccc3)c3ccccc3)CC2)cc(C)n1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
KDM4E B2RXH2 3/20 0.47
MAPT P10636 1/20 0.47
LMNA P02545 3/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HTT P42858 1/20 0.46
HIF1A Q16665 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
POLB P06746 1/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
TSHR P16473 1/20 0.45
GAA P10253 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
CYP2D6 P10635 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4271755 0.93 LMNA (0.46) ALDH1A1CYP3A4CYP2C9KDM4EMAPT
SCHEMBL5065803 0.85 LMNA (0.58) ALDH1A1LMNASMN1; SMN2HTTPOLB
SCHEMBL10335011 0.81 MEN1 (0.57) ALDH1A1CYP3A4HIF1APOLBMEN1
SCHEMBL4279870 0.79 ALDH1A1 (0.52) ALDH1A1CYP3A4CYP2C9KDM4EMAPT
SCHEMBL4271439 0.74 DRD2 (0.46) ALDH1A1KDM4EMAPTLMNASMN1; SMN2
SCHEMBL4275831 0.74 NPC1 (0.71) ALDH1A1CYP3A4KMT2ANPC1CYP2D6
SCHEMBL4275876 0.71 CACNA2D1 (0.73) TDP1POLBCYP2D6
SCHEMBL4278641 0.71 CA12 (0.46) ALDH1A1CYP3A4CYP2C9KDM4EMAPT
SCHEMBL1088276 0.71 CYP2D6 (0.78) ALDH1A1CYP3A4CYP2C9KDM4ELMNA
SCHEMBL11374977 0.71 LMNA (0.70) ALDH1A1CYP3A4CYP2C9KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007071035-A1 HETEROCYCLIC AMIDE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS NEUROMED PHARMACEUTICALS LTD. (CA) 2007-06-28 WO disclosed