SCHEMBL8237608

SCHEMBL8237608

C=C(COC(c1ccccc1)c1ccccc1)N1C(C)CN(CC2CCOCC2)CC1C

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
TACR2 P21452 1/20 0.38
MAPK1 P28482 1/20 0.38
SLC6A4 P31645 2/20 0.36
SLC6A3 Q01959 2/20 0.36
SLC6A2 P23975 1/20 0.36
CACNA1G O43497 1/20 0.36
CACNA1H O95180 1/20 0.36
PRKCB P05771 1/20 0.36
CYP3A4 P08684 1/20 0.35
HTR4 Q13639 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4275673 0.87 TACR2 (0.46) SIGMAR1KDM4EALDH1A1POLBTACR2
SCHEMBL4271169 0.74 TACR2 (0.43) ALDH1A1TACR2CACNA1GCACNA1HPRKCB
SCHEMBL4279734 0.73 TACR2 (0.60) KDM4EALDH1A1POLBTACR2SLC6A4
SCHEMBL5047955 0.73 CACNA1G (0.39) SIGMAR1KDM4EALDH1A1POLBTACR2
SCHEMBL4272230 0.72 TACR2 (0.42) TACR2SLC6A3CACNA1GCACNA1HCYP3A4
SCHEMBL5048006 0.66 CACNA1G (0.38) TACR2CACNA1GCACNA1HPRKCBCYP3A4
SCHEMBL2794338 0.66 CACNA2D1 (0.50) ALDH1A1TACR2SLC6A4SLC6A3SLC6A2
SCHEMBL5051949 0.65 TACR2 (0.37) TACR2CACNA1GCACNA1HPRKCBCYP3A4
SCHEMBL5053752 0.65 GRM5 (0.38) POLBTACR2MAPK1SLC6A3SLC6A2
SCHEMBL2794421 0.62 CACNA2D1 (0.66) ALDH1A1POLBSLC6A4SLC6A3SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007071035-A1 HETEROCYCLIC AMIDE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS NEUROMED PHARMACEUTICALS LTD. (CA) 2007-06-28 WO disclosed