SCHEMBL8238176

SCHEMBL8238176

COc1ccc2c(c1)nc(C)n2-c1cnc(NC(=O)c2ccc(C#N)cc2)cn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
USP2 O75604 1/20 0.47
LMNA P02545 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
HPGD P15428 2/20 0.44
HSD17B10 Q99714 2/20 0.43
HSP90AA1 P07900 1/20 0.43
HSP90AB1 P08238 1/20 0.43
GSK3B P49841 2/20 0.43
DYRK1A Q13627 2/20 0.43
ITK Q08881 3/20 0.43
THRB P10828 2/20 0.43
ADORA2A P29274 1/20 0.42
GCK P35557 1/20 0.42
KCNH2 Q12809 1/20 0.42
DEGS1 O15121 2/20 0.41
HDAC4 P56524 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HPGDS O60760 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8238174 0.89 RAB9A (0.48) ALDH1A1LMNANPSR1HSD17B10HSP90AA1
SCHEMBL648227 0.88 HDAC4 (0.48) ALDH1A1USP2LMNANPSR1L3MBTL1
SCHEMBL8234112 0.87 TP53 (0.45) ALDH1A1HPGDHSD17B10HSP90AA1HSP90AB1
SCHEMBL8234439 0.86 TP53 (0.45) ALDH1A1HPGDHSD17B10HSP90AA1HSP90AB1
SCHEMBL8233770 0.85 TP53 (0.43) ALDH1A1HPGDHSD17B10HSP90AA1HSP90AB1
SCHEMBL8236747 0.83 NPC1 (0.46) ALDH1A1LMNAHPGDHSD17B10HSP90AA1
SCHEMBL8234043 0.83 PLK1 (0.48) LMNAHSD17B10HSP90AA1HSP90AB1THRB
SCHEMBL8234051 0.80 ALOX15 (0.49) NPSR1L3MBTL1HSD17B10THRBMAPK1
SCHEMBL3103400 0.80 RAB9A (0.45) LMNAHSD17B10HSP90AA1HSP90AB1THRB
SCHEMBL8236417 0.80 RAB9A (0.51) LMNANPSR1HPGDHSD17B10HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007109362-A2 BENZOIMIDAZOLYL-PARAZINE COMPOUNDS FOR INFLAMMATION AND IMMUNE-RELATED USES SYNTA PHARMACEUTICALS CORP. (US) 2007-09-27 WO disclosed