SCHEMBL8238538

SCHEMBL8238538

Nc1ccc(-c2ccc(F)c(F)c2)nc1N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 2/20 0.44
ALDH1A1 P00352 3/20 0.41
CYP1A2 P05177 1/20 0.41
GAA P10253 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
KLK7 P49862 1/20 0.40
TRPV3 Q8NET8 1/20 0.40
HDAC2 Q92769 1/20 0.38
RAB9A P51151 4/20 0.38
NPC1 O15118 3/20 0.38
MAP4K4 O95819 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
MINK1 Q8N4C8 2/20 0.38
TNIK Q9UKE5 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPK1 P28482 1/20 0.38
TP53 P04637 1/20 0.38
PKM P14618 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31224683 0.75 NPC1 (0.48) ALDH1A1CYP1A2GAACYP2C9CYP2C19
SCHEMBL1463746 0.75 MAPT (0.47) KMOALDH1A1CYP1A2GAACYP2C9
SCHEMBL21200228 0.73 ALDH1A1 (0.54) ALDH1A1HDAC2MAP4K4MAPK1HSD17B10
SCHEMBL898443 0.73 ALDH1A1 (0.45) ALDH1A1NPC1MPL
SCHEMBL30873896 0.71 SMN1; SMN2 (0.44) ALDH1A1CYP1A2CYP2C9CYP2C19RAB9A
SCHEMBL30738324 0.71 ALDH1A1 (0.50) ALDH1A1CYP1A2GAACYP2C9CYP2C19
SCHEMBL22179700 0.71 ALDH1A1 (0.50) ALDH1A1CYP1A2GAACYP2C9CYP2C19
SCHEMBL24067959 0.71 LMNA (0.42) ALDH1A1GAARAB9ANPC1MAP4K4
SCHEMBL126685 0.70 MPL (0.69) ALDH1A1RAB9ANPC1SMN1; SMN2KDM4E
SCHEMBL4053052 0.70 MAP2K3 (0.56) ALDH1A1RAB9ANPC1SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007020521-A1 PYRIDOYRAZINONES AS PDE-5 INHIBITORS PHARMACIA & UPJOHN COMPANY LLC (US) 2007-02-22 WO disclosed