SCHEMBL898443

SCHEMBL898443

Nc1ccc(-c2cc(F)ccc2F)nc1N

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.45
NPC1 O15118 1/20 0.38
MPL P40238 1/20 0.36
ADORA2A P29274 2/20 0.36
ADORA1 P30542 2/20 0.36
CCNE1 P24864 2/20 0.35
CDK2 P24941 2/20 0.35
CDC7 O00311 1/20 0.35
DBF4 Q9UBU7 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CASP3 P42574 1/20 0.35
SENP8 Q96LD8 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
SENP6 Q9GZR1 1/20 0.35
SLC9A1 P19634 1/20 0.35
IL4 P05112 1/20 0.35
BACE1 P56817 1/20 0.34
KEAP1 Q14145 1/20 0.34
LMNA P02545 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2884296 0.86 ALDH1A1 (0.50) ALDH1A1MPLADORA2AADORA1
SCHEMBL1582795 0.78 MPL (0.53) ALDH1A1NPC1MPLADORA2AL3MBTL1
SCHEMBL4402521 0.73 L3MBTL1 (0.42) NPC1L3MBTL1CASP3SENP8SENP7
SCHEMBL8238538 0.73 KMO (0.44) ALDH1A1NPC1MPL
SCHEMBL1582458 0.72 NPC1 (0.39) ALDH1A1NPC1CCNE1CDK2CDC7
SCHEMBL14018473 0.71 KDM1A (0.44) ALDH1A1MPLCCNE1CDK2CDC7
SCHEMBL31006087 0.71 MPL (0.67) ALDH1A1NPC1MPLLMNAHTT
SCHEMBL1916792 0.71 MPL (0.67) ALDH1A1NPC1MPLLMNAHTT
SCHEMBL2596804 0.71 AGPAT2 (0.39) ALDH1A1NPC1MPLCCNE1CDK2
SCHEMBL25375541 0.69 ABL1 (0.41) ALDH1A1SLC9A1LMNAAGPAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed