SCHEMBL8244272

SCHEMBL8244272

O=Cc1ccc2c(c1)CNCCS2

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RYR2 Q92736 3/20 0.55
KCNH2 Q12809 1/20 0.55
CYP2A6 P11509 3/20 0.34
ALDH1A1 P00352 4/20 0.33
MEN1 O00255 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B10 Q99714 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
KDM4E B2RXH2 1/20 0.32
PTGS2 P35354 1/20 0.32
RAB9A P51151 1/20 0.32
PNMT P11086 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4824838 0.78 ALDH1A1 (0.40) CYP2A6ALDH1A1MEN1GAAMAPT
SCHEMBL10366338 0.75 ALDH1A1 (0.45) CYP2A6ALDH1A1MEN1GAAMAPT
SCHEMBL28461427 0.75 RYR2 (0.59) RYR2KCNH2MAPTKDM4EPNMT
SCHEMBL2600211 0.75 RYR2 (0.64) RYR2KCNH2MEN1MAPTKMT2A
SCHEMBL8134941 0.75 RYR2 (0.59) RYR2KCNH2ALDH1A1MEN1GAA
SCHEMBL2062318 0.75 RYR2 (0.59) RYR2KCNH2ALDH1A1MEN1GAA
SCHEMBL14691898 0.75 RYR2 (0.59) RYR2KCNH2ALDH1A1MEN1GAA
SCHEMBL16976367 0.74 RYR2 (0.55) RYR2KCNH2ALDH1A1MEN1GAA
SCHEMBL3054155 0.73 ALDH1A1 (0.49) RYR2KCNH2CYP2A6ALDH1A1MEN1
SCHEMBL3944638 0.73 ASIC3 (0.55) PNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007024717-A2 AGENTS FOR PREVENTING AND TREATING DISORDERS INVOLVING MODULATION OF THE RYR RECEPTORS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2007-03-01 WO disclosed