SCHEMBL8246744

SCHEMBL8246744

Cc1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)NCc2ccccc2)o1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.51
NPSR1 Q6W5P4 1/20 0.51
HPGD P15428 3/20 0.50
LMNA P02545 1/20 0.49
MAPK1 P28482 1/20 0.49
POLB P06746 2/20 0.48
MMP2 P08253 1/20 0.48
PSMB5 P28074 3/20 0.47
NFKB1 P19838 2/20 0.47
NFKB2 Q00653 2/20 0.47
RELA Q04206 2/20 0.47
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA3 P07451 1/20 0.45
CA4 P22748 1/20 0.45
CA6 P23280 1/20 0.45
CA5A P35218 1/20 0.45
CA7 P43166 1/20 0.45
CACNA1C Q13936 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3577956 0.86 KDM4E (0.55) ALDH1A1NPSR1HPGDLMNAMAPK1
SCHEMBL3581117 0.86 HPGD (0.62) ALDH1A1NPSR1HPGDLMNAPOLB
SCHEMBL3581142 0.84 MMP2 (0.47) ALDH1A1HPGDLMNAMMP2PSMB5
SCHEMBL3578207 0.81 MMP2 (0.46) ALDH1A1HPGDLMNAMAPK1MMP2
SCHEMBL7741059 0.81 MMP2 (0.54) POLBMMP2PSMB5NFKB1NFKB2
SCHEMBL7741064 0.81 MMP2 (0.54) POLBMMP2PSMB5NFKB1NFKB2
SCHEMBL3588641 0.80 RAB9A (0.48) ALDH1A1NPSR1HPGDLMNAMAPK1
SCHEMBL2246985 0.78 ADAMTS5 (0.59) MMP2PSMB5NFKB1NFKB2RELA
SCHEMBL3576509 0.78 ADAMTS5 (0.62) MAPK1MMP2MMP8
SCHEMBL3581169 0.78 C3AR1 (0.57) ALDH1A1HPGDMMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007008994-A2 GLUTAMATE AGGRECANASE INHIBITORS WYETH (US) 2007-01-18 WO disclosed