SCHEMBL8248232

SCHEMBL8248232

COC(=O)C1CCC(C(=O)Nc2sc3c(c2C(=O)NCCc2ccccc2)CCCC3)CC1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 6/20 0.65
CNR1 P21554 1/20 0.65
TAAR1 Q96RJ0 2/20 0.58
MAPT P10636 2/20 0.57
KDM4E B2RXH2 2/20 0.57
HSD17B10 Q99714 1/20 0.57
KMT2A Q03164 3/20 0.56
MEN1 O00255 2/20 0.56
ALDH1A1 P00352 2/20 0.56
SMN1; SMN2 Q16637 1/20 0.53
ATM Q13315 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
RORC P51449 2/20 0.52
FLT3 P36888 1/20 0.51
NPC1 O15118 1/20 0.51
TP53 P04637 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7886940 0.92 TAAR1 (0.61) CNR2CNR1TAAR1MAPTKDM4E
SCHEMBL8206909 0.91 RORC (0.63) CNR2CNR1MAPTKDM4EHSD17B10
Bicarbonate SCHEMBL7886942 0.90 CNR2 (0.66) CNR2CNR1TAAR1MAPTKDM4E
SCHEMBL8212606 0.82 CNR2 (0.61) CNR2CNR1MAPTKDM4EHSD17B10
SCHEMBL7890904 0.82 RORC (0.67) CNR2CNR1MAPTKDM4EHSD17B10
SCHEMBL8206447 0.81 KMT2A (0.66) CNR2TAAR1MAPTKMT2AMEN1
SCHEMBL3801324 0.81 RORC (0.68) CNR2CNR1MAPTKDM4EALDH1A1
SCHEMBL8248235 0.80 MAPT (0.58) CNR2CNR1MAPTKDM4EHSD17B10
SCHEMBL8200351 0.80 CNR2 (0.54) CNR2CNR1MAPTKDM4EHSD17B10
SCHEMBL8207571 0.80 CNR2 (0.58) CNR2CNR1MAPTKDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6143777-A ENZYME INHIBITORS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-07 US disclosed