SCHEMBL8249461

SCHEMBL8249461

C=CCOc1ccc2ccnc(O)c2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.44
CA1 P00915 4/20 0.44
CA9 Q16790 4/20 0.44
MAOA P21397 2/20 0.44
MTNR1A P48039 2/20 0.44
MAPT P10636 2/20 0.43
LMNA P02545 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
HPGD P15428 3/20 0.41
ALDH1A1 P00352 2/20 0.41
GAA P10253 2/20 0.41
ADRA2A P08913 1/20 0.39
ADRA2B P18089 1/20 0.39
ADRA2C P18825 1/20 0.39
KDM4E B2RXH2 1/20 0.38
POLB P06746 1/20 0.38
PKM P14618 1/20 0.38
ALDH2 P05091 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1244080 0.82 CA12 (0.44) CA12CA1CA9MAOAMTNR1A
SCHEMBL20537232 0.77 MTNR1A (0.53) CA12CA1CA9MTNR1AMAPT
SCHEMBL3825460 0.76 CA12 (0.64) CA12CA1CA9MAOAMTNR1A
SCHEMBL12055259 0.76 PLAU (0.59) MTNR1ALMNAKDM4ENPSR1PLAU
SCHEMBL8477878 0.74 CA12 (0.54) CA12CA1CA9MAOAMAPT
SCHEMBL7650010 0.73 CA12 (0.57) CA12CA1CA9MAOAMTNR1A
SCHEMBL3823460 0.73 CA12 (0.60) CA12CA1CA9MAPTLMNA
SCHEMBL3824435 0.72 MTNR1A (0.51) CA12CA1CA9MTNR1AMAPT
SCHEMBL31299883 0.72 ABL1 (0.40) MAPTALDH1A1GAAKDM4EPLAU
SCHEMBL29576500 0.72 LTA4H (0.44) PLAUPLAT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007016441-A1 MACROCYCLIC PEPTIDES AS HCV NS3 PROTEASE INHIBITORS MERCK & CO., INC. (US) 2007-02-08 WO disclosed