SCHEMBL8250274

SCHEMBL8250274

COc1ccc2c(c1)CN(CCC(=O)O)C2=O

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.60
ALOX15 P16050 1/20 0.60
TSHR P16473 1/20 0.60
SIRT1 Q96EB6 1/20 0.60
ITGB3 P05106 6/20 0.57
ITGAV P06756 3/20 0.57
ADAM17 P78536 2/20 0.51
ITGA2B P08514 3/20 0.47
KMO O15229 1/20 0.46
ALDH1A1 P00352 1/20 0.45
HPGD P15428 1/20 0.45
PRMT5 O14744 1/20 0.45
WDR77 Q9BQA1 1/20 0.45
METAP1 P53582 1/20 0.43
AOC3 Q16853 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8049969 0.84 ADAM17 (0.44) KDM4EALOX15TSHRSIRT1ITGB3
SCHEMBL6440847 0.82 ADAM17 (0.51) KDM4EADAM17ALDH1A1PRMT5WDR77
SCHEMBL8547905 0.79 ADAM17 (0.53) KDM4EADAM17ALDH1A1PRMT5WDR77
SCHEMBL15776135 0.78 ADAM17 (0.44) KDM4EALOX15TSHRSIRT1ITGB3
SCHEMBL1002943 0.77 ADAM17 (0.57) KDM4EADAM17ALDH1A1PRMT5WDR77
SCHEMBL22446339 0.77 HDAC6 (0.45) ADAM17AOC3
SCHEMBL7788827 0.76 ITGB3 (0.69) ITGB3ITGA2BAOC3
SCHEMBL15169553 0.76 METAP1 (0.45) KDM4EADAM17ALDH1A1HPGDPRMT5
SCHEMBL22713735 0.76 AOC3 (0.69) ITGB3ITGAVITGA2BPRMT5WDR77
SCHEMBL315339 0.76 KDM4E (1.00) KDM4EALOX15TSHRSIRT1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007001249-A1 NITROGEN HETEROCYCLE BIARYLS FOR OSTEOPOROSIS AND OTHER DISEASES PHARMACOPEIA, INC. (US) 2007-01-04 WO disclosed