SCHEMBL8250573

SCHEMBL8250573

CS(=O)(=O)Nc1ccccc1N1CCN(C(=O)c2cccnc2F)CC1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
KDM4E B2RXH2 2/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
TSHR P16473 2/20 0.48
GPR6 P46095 2/20 0.46
NPY5R Q15761 1/20 0.45
LMNA P02545 5/20 0.45
MAPT P10636 2/20 0.45
EED O75530 1/20 0.44
GAA P10253 2/20 0.43
GLA P06280 1/20 0.43
NPC1 O15118 1/20 0.43
TP53 P04637 1/20 0.43
HTT P42858 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8240451 0.82 ALDH1A1 (0.60) ALDH1A1SMN1; SMN2KDM4EL3MBTL1TSHR
SCHEMBL8239707 0.79 ALDH1A1 (0.46) ALDH1A1TSHRGPR6MAPTGAA
SCHEMBL8247932 0.78 ALDH1A1 (0.63) ALDH1A1KDM4EL3MBTL1TSHRMAPT
SCHEMBL4721325 0.77 HSD11B1 (0.59) ALDH1A1SMN1; SMN2KDM4EL3MBTL1TSHR
SCHEMBL4524859 0.76 NPY5R (0.52) ALDH1A1SMN1; SMN2KDM4ETSHRNPY5R
SCHEMBL4721446 0.74 GAA (0.59) ALDH1A1SMN1; SMN2KDM4EL3MBTL1TSHR
SCHEMBL4766135 0.72 USP2 (0.57) ALDH1A1SMN1; SMN2KDM4EL3MBTL1TSHR
SCHEMBL8247070 0.72 SMN1; SMN2 (0.72) ALDH1A1SMN1; SMN2KDM4EL3MBTL1TSHR
SCHEMBL4513123 0.71 NPY5R (0.48) ALDH1A1SMN1; SMN2NPY5RLMNAMAPT
SCHEMBL14355835 0.71 TSHR (0.52) ALDH1A1SMN1; SMN2TSHRLMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007009635-A1 PHENYL SUBSTITUTED PIPERAZINE-DERIVATIVES AS INHIBITORS OF PLAMINOGENIC ACTIVATOR INHIBITORS-I (PAI-I) BAYER HEALTHCARE AG (DE) 2007-01-25 WO disclosed