SCHEMBL8240451

SCHEMBL8240451

O=C(c1cccnc1F)N1CCN(c2ccccc2Cl)CC1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.60
KDM4E B2RXH2 3/20 0.60
HSD17B10 Q99714 3/20 0.60
HPGD P15428 1/20 0.60
MAPT P10636 4/20 0.58
MEN1 O00255 2/20 0.58
KMT2A Q03164 2/20 0.58
SMN1; SMN2 Q16637 4/20 0.57
TSHR P16473 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.56
GAA P10253 1/20 0.56
POLB P06746 1/20 0.52
PKM P14618 1/20 0.52
MAPK1 P28482 1/20 0.51
RAB9A P51151 1/20 0.51
LMNA P02545 3/20 0.51
P2RX7 Q99572 1/20 0.49
RBP4 P02753 1/20 0.49
AVPR1A P37288 1/20 0.49
USP2 O75604 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4721446 0.91 GAA (0.59) ALDH1A1KDM4EHSD17B10HPGDMAPT
SCHEMBL4721325 0.84 HSD11B1 (0.59) ALDH1A1KDM4ESMN1; SMN2TSHRL3MBTL1
SCHEMBL8247932 0.83 ALDH1A1 (0.63) ALDH1A1KDM4EHSD17B10MAPTMEN1
SCHEMBL4722869 0.82 AKR1C3 (0.58) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL4718989 0.82 ALDH1A1 (0.53) ALDH1A1KDM4EHSD17B10HPGDMAPT
SCHEMBL8250573 0.82 ALDH1A1 (0.48) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL4719103 0.81 ABL1 (0.55) ALDH1A1KDM4EHSD17B10HPGDMAPT
SCHEMBL8247070 0.79 SMN1; SMN2 (0.72) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL23064276 0.78 GAA (0.67) ALDH1A1KDM4EHSD17B10HPGDMAPT
SCHEMBL9565871 0.78 SMN1; SMN2 (0.57) ALDH1A1KDM4EHSD17B10HPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007009635-A1 PHENYL SUBSTITUTED PIPERAZINE-DERIVATIVES AS INHIBITORS OF PLAMINOGENIC ACTIVATOR INHIBITORS-I (PAI-I) BAYER HEALTHCARE AG (DE) 2007-01-25 WO disclosed