SCHEMBL8250811

SCHEMBL8250811

Cc1noc(-c2ccc(Br)cc2)c1/C(O)=C/O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.36
NR1H4 Q96RI1 1/20 0.34
ALDH1A1 P00352 3/20 0.34
MAPT P10636 3/20 0.34
RXFP1 Q9HBX9 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
KDM4E B2RXH2 1/20 0.34
POLB P06746 1/20 0.34
PKM P14618 1/20 0.34
TRPV1 Q8NER1 1/20 0.33
RAB9A P51151 1/20 0.33
TP53 P04637 1/20 0.33
PTGS1 P23219 1/20 0.33
NPC1 O15118 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
LPAR1 Q92633 1/20 0.32
LPAR3 Q9UBY5 1/20 0.32
EDNRB P24530 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1563 0.81 PTPN1 (0.47) PTPN1ALDH1A1MAPTRXFP1MEN1
SCHEMBL1784 0.77 ALDH1A1 (0.40) PTPN1ALDH1A1MAPTRXFP1MEN1
SCHEMBL4233 0.77 BACE1 (0.44) ALDH1A1MAPTSMN1; SMN2KDM4EPOLB
SCHEMBL1883 0.75 RAB9A (0.57) ALDH1A1MAPTMEN1KMT2ASMN1; SMN2
SCHEMBL1447 0.75 GSK3B (0.42) PTPN1ALDH1A1MAPTRXFP1SMN1; SMN2
SCHEMBL27886960 0.73 EDNRB (0.45) NR1H4ALDH1A1MAPTMEN1KMT2A
SCHEMBL8243211 0.72 ALDH1A1 (0.64) ALDH1A1MAPTRXFP1MEN1KMT2A
SCHEMBL1736 0.72 NR1H4 (0.35) NR1H4ALDH1A1MAPTMEN1KMT2A
SCHEMBL22480523 0.71 NPC1 (0.46) PTPN1ALDH1A1MAPTSMN1; SMN2KDM4E
Benzene SCHEMBL13719765 0.71 ALDH1A1 (0.36) PTPN1ALDH1A1MAPTRXFP1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007002214-A2 ACYL GUANIDINES AS BETA-SECRETASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-01-04 WO disclosed