SCHEMBL8258604

SCHEMBL8258604

O=c1c(Cl)c(CN2CCN(c3ncc(C(F)(F)F)cc3Cl)CC2)[nH]n1-c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
GRM2 Q14416 2/20 0.52
DRD2 P14416 1/20 0.52
DRD4 P21917 1/20 0.52
DRD3 P35462 1/20 0.52
SMN1; SMN2 Q16637 5/20 0.50
MAPT P10636 5/20 0.50
ALDH1A1 P00352 3/20 0.50
NPSR1 Q6W5P4 1/20 0.50
CHRM4 P08173 3/20 0.49
LMNA P02545 2/20 0.47
HTT P42858 2/20 0.47
TSHR P16473 1/20 0.47
KDM4E B2RXH2 1/20 0.47
POLB P06746 1/20 0.47
HPGD P15428 1/20 0.47
CHRM5 P08912 1/20 0.47
CHRM1 P11229 1/20 0.47
CHRM3 P20309 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4318192 0.80 GRM2 (0.57) MEN1KMT2AGRM2DRD2DRD4
SCHEMBL2675769 0.74 MEN1 (0.52) MEN1KMT2AGRM2DRD2DRD4
SCHEMBL4318159 0.73 ALDH1A1 (0.48) MEN1KMT2ADRD2DRD4DRD3
SCHEMBL8255009 0.73 ALDH1A1 (0.47) MEN1KMT2ADRD2DRD4DRD3
SCHEMBL4244132 0.72 MEN1 (0.56) MEN1KMT2AGRM2DRD2DRD4
SCHEMBL5199448 0.71 DRD2 (0.55) MEN1KMT2AGRM2DRD2DRD4
SCHEMBL4166695 0.69 MEN1 (0.60) MEN1KMT2AGRM2DRD2DRD4
Bromide SCHEMBL4174809 0.69 MEN1 (0.59) MEN1KMT2AGRM2DRD2DRD4
SCHEMBL24606221 0.69 GRM2 (1.00) MEN1KMT2AGRM2DRD2DRD4
SCHEMBL29709278 0.69 GRM2 (1.00) MEN1KMT2AGRM2DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006071730-A1 PYRAZOLONE COMPOUNDS AS METABOTROPIC GLUTAMATE RECEPTOR AGONISTS FOR THE TREATMENT OF NEUROLOGICAL AND PSYCHIATRIC DISORDERS ASTRAZENECA AB (SE) 2006-07-06 WO disclosed