SCHEMBL8260306

SCHEMBL8260306

CCCN(CC(=O)Nc1ccc2sc(C(=O)NO)cc2c1)C(=O)COc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 12/20 0.55
NPC1 O15118 1/20 0.46
MAPT P10636 3/20 0.46
RAB9A P51151 1/20 0.45
PSMB5 P28074 1/20 0.45
POLB P06746 1/20 0.44
GAA P10253 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5809271 0.84 HDAC1 (0.71) HDAC1NPC1MAPTRAB9APOLB
SCHEMBL8258697 0.83 HDAC1 (0.63) HDAC1
SCHEMBL8257248 0.80 HDAC1 (0.60) HDAC1L3MBTL1
SCHEMBL8260320 0.78 HDAC1 (0.67) HDAC1NPC1MAPTRAB9A
SCHEMBL5805572 0.74 HDAC1 (0.71) HDAC1RAB9A
SCHEMBL5808017 0.73 HDAC1 (0.62) HDAC1NPC1MAPTRAB9APOLB
SCHEMBL8257257 0.72 HDAC1 (0.51) HDAC1MAPT
SCHEMBL1893680 0.72 HDAC1 (1.00) HDAC1
SCHEMBL5805563 0.72 HDAC1 (0.73) HDAC1
SCHEMBL8291158 0.72 HDAC1 (0.69) HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006101454-A1 BENZOTHIOPHENE DERIVATIVES: PREPARATION AND PHARMACEUTICAL APPLICATIONS S*BIO PTE LTD (SG) 2006-09-28 WO disclosed