SCHEMBL8265602

SCHEMBL8265602

C=C(CSC(C)=O)c1ccc(CN(C)c2ccc(OC)cc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 3/20 0.52
HDAC4 P56524 3/20 0.52
HDAC1 Q13547 3/20 0.52
HDAC7 Q8WUI4 3/20 0.52
HDAC2 Q92769 3/20 0.52
HDAC10 Q969S8 3/20 0.52
HDAC11 Q96DB2 3/20 0.52
HDAC8 Q9BY41 3/20 0.52
HDAC6 Q9UBN7 3/20 0.52
HDAC9 Q9UKV0 3/20 0.52
HDAC5 Q9UQL6 3/20 0.52
CNR1 P21554 1/20 0.46
CNR2 P34972 1/20 0.46
ACHE P22303 1/20 0.44
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
ALDH1A1 P00352 2/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TSPO P30536 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4880423 0.88 HDAC3 (0.70) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL19302284 0.76 PYCR1 (0.53) ACHEMEN1KMT2AALDH1A1HTT
SCHEMBL4880366 0.70 HDAC3 (0.74) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL12526817 0.70 ACHE (0.54) CNR1CNR2ACHEALDH1A1HTT
SCHEMBL29336359 0.69 MEN1 (0.50) MEN1KMT2AALDH1A1HTTSMN1; SMN2
SCHEMBL29336627 0.69 BCL2A1 (0.56) HDAC1CNR2ALDH1A1HTTSMN1; SMN2
SCHEMBL14266667 0.68 TSHR (0.57) CNR1CNR2ACHEALDH1A1LMNA
SCHEMBL19057672 0.68 LTA4H (0.55) CNR1CNR2ACHEMEN1KMT2A
SCHEMBL4883456 0.68 HDAC3 (0.80) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL5320248 0.67 HDAC3 (0.78) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006063294-A2 NOVEL INHIBITORS OF HISTONE DEACETYLASE FOR THE TREATMENT OF DISEASE KALYPSYS, INC. (US) 2006-06-15 WO disclosed