SCHEMBL8268409

SCHEMBL8268409

Cc1cc2ccc(I)cc2s1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
APP P05067 2/20 0.36
ALDH1A1 P00352 1/20 0.34
DHPS P49366 1/20 0.34
ESR1 P03372 3/20 0.33
ESR2 Q92731 3/20 0.33
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC10 Q969S8 1/20 0.33
HDAC11 Q96DB2 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
HDAC9 Q9UKV0 1/20 0.33
HDAC5 Q9UQL6 1/20 0.33
MAPT P10636 1/20 0.33
CHRNA7 P36544 1/20 0.32
TYMS P04818 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8291879 0.83 CYP2A6 (0.36) APPALDH1A1
SCHEMBL422041 0.77 HDAC3 (0.52) APPALDH1A1ESR1ESR2HDAC3
SCHEMBL2091131 0.74 DHPS (0.34) APPDHPS
SCHEMBL31009687 0.74 CYP2A6 (0.38) APPALDH1A1HDAC3HDAC4HDAC1
SCHEMBL3962610 0.74 CYP2A6 (0.38) APPALDH1A1HDAC3HDAC4HDAC1
SCHEMBL147786 0.74 GFER (0.41) APPALDH1A1MAPTCHRNA7
SCHEMBL12278184 0.74 CA2 (0.52) APPALDH1A1MAPT
SCHEMBL5241572 0.74 ESR2 (0.58) ESR1ESR2
SCHEMBL144486 0.74 ALDH1A1 (0.38) ALDH1A1ESR1ESR2MAPTCHRNA7
SCHEMBL2742924 0.73 ALDH1A1 (0.38) ALDH1A1HDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006041831-A2 CYCLIC Β-AMINO ACID DERIVATIVES AS FACTOR XA INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2006-04-20 WO disclosed
WO-2005032468-A2 MONOCYCLIC AND BICYCLIC LACTAMS AS FACTOR XA INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2005-04-14 WO disclosed
WO-2003026652-A1 LACTAM-CONTAINING COMPOUNDS AND DERIVATIVES THEREOF AS FACTOR XA INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-04-03 WO disclosed