SCHEMBL8272191

SCHEMBL8272191

CC(O)CCN(c1ccc(Cl)cc1C(O)c1ccccc1Cl)S(=O)(=O)c1ccc2c(c1)OC(C)O2

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
FDFT1 P37268 16/20 0.39
ESR1 P03372 2/20 0.35
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
APH1B Q8WW43 1/20 0.35
NCSTN Q92542 1/20 0.35
APH1A Q96BI3 1/20 0.35
PSENEN Q9NZ42 1/20 0.35
RORC P51449 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8272192 0.91 FDFT1 (0.40) FDFT1ESR1PSEN1PSEN2APH1B
SCHEMBL8272847 0.88 FDFT1 (0.41) FDFT1
SCHEMBL8272193 0.85 FDFT1 (0.47) FDFT1
SCHEMBL8275043 0.82 FDFT1 (0.36) FDFT1
SCHEMBL8272194 0.81 FDFT1 (0.35) FDFT1
SCHEMBL8272196 0.77 TP53 (0.40) FDFT1
SCHEMBL8272848 0.76 PKM (0.44) FDFT1
SCHEMBL3252395 0.74 KEAP1 (0.52) FDFT1
SCHEMBL4872059 0.74 KEAP1 (0.52) FDFT1
SCHEMBL3253822 0.73 PKM (0.49) FDFT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1776347-B1 SULPHONAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION SANOFI AVENTIS (FR) 2010-05-26 EP disclosed
WO-2006024779-A1 SULPHONAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION SANOFI-AVENTIS (FR) 2006-03-09 WO disclosed