SCHEMBL8273095

SCHEMBL8273095

COc1nccc2c(OC)c(Cl)ccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.39
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 2/20 0.37
HSD17B10 Q99714 1/20 0.37
CYP2C19 P33261 2/20 0.35
CYP1A2 P05177 1/20 0.35
DYRK1A Q13627 3/20 0.35
PDE1B Q01064 2/20 0.34
PDE2A O00408 1/20 0.34
PDE8B O95263 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
HTR2B P41595 1/20 0.34
PDE1A P54750 1/20 0.34
PDE4D Q08499 1/20 0.34
PDE1C Q14123 1/20 0.34
PDE11A Q9HCR9 1/20 0.34
PDE10A Q9Y233 1/20 0.34
MAPK1 P28482 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MAPT P10636 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13409351 0.85 LRRK2 (0.36) MAOAALDH1A1KDM4EHSD17B10CYP2C19
SCHEMBL1536585 0.84 MAPK1 (0.44) MAOAALDH1A1KDM4EHSD17B10CYP2C19
SCHEMBL8271693 0.80 CYP2C19 (0.43) MAOAALDH1A1KDM4EHSD17B10CYP2C19
SCHEMBL8272295 0.76 CYP1A2 (0.48) ALDH1A1KDM4EHSD17B10CYP2C19CYP1A2
SCHEMBL12780743 0.75 CYP19A1 (0.48) ALDH1A1CYP2C19CYP1A2DYRK1APDE1B
SCHEMBL2239481 0.74 TRPA1 (0.37) ALDH1A1CYP2C19CYP1A2DYRK1AMAPK1
SCHEMBL30666115 0.70 KDM4E (0.40) MAOAALDH1A1KDM4EHSD17B10CYP1A2
SCHEMBL26656449 0.70 KDM4E (0.40) MAOAALDH1A1KDM4EHSD17B10CYP1A2
SCHEMBL911419 0.69 CCR4 (0.43) DYRK1AMAPK1MAPTNFE2L2GRM4
SCHEMBL11755564 0.69 ALDH1A1 (0.39) MAOAALDH1A1KDM4EHSD17B10DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006000085-A1 HEPATITIS C INHIBITOR PEPTIDE ANALOGS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2006-01-05 WO disclosed