SCHEMBL13409351

SCHEMBL13409351

COc1c(Cl)ccc2c(OC(C)C)nccc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.36
MAOA P21397 1/20 0.34
ATM Q13315 2/20 0.33
MAPT P10636 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
TRPM8 Q7Z2W7 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ADRA2A P08913 2/20 0.32
ADRA2B P18089 2/20 0.32
ADRA2C P18825 2/20 0.32
ADRA1A P35348 2/20 0.32
HTR1A P08908 1/20 0.32
SLC6A4 P31645 1/20 0.32
OPRK1 P41145 1/20 0.32
KCNH2 Q12809 1/20 0.32
PDE1B Q01064 2/20 0.32
RORC P51449 1/20 0.32
PDE2A O00408 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8273095 0.85 MAOA (0.39) MAOAMAPTKDM4EALDH1A1HSD17B10
SCHEMBL13409342 0.83 PDE1B (0.39) LRRK2MAOAMAPTTRPM8KDM4E
SCHEMBL13409340 0.79 CYP19A1 (0.43) LRRK2MAPTL3MBTL1TRPM8PDE1B
SCHEMBL1536585 0.77 MAPK1 (0.44) MAOAMAPTKDM4EALDH1A1HSD17B10
SCHEMBL13409336 0.76 ATM (0.44) LRRK2ATMMAPTL3MBTL1KDM4E
SCHEMBL13409320 0.72 PLAU (0.49) LRRK2ATMMAPTTRPM8KDM4E
SCHEMBL13409346 0.72 LRRK2 (0.38) LRRK2ATMMAPTTRPM8CYP2C19
SCHEMBL31701118 0.71 LRRK2 (0.40) LRRK2ATMMAPTL3MBTL1KDM4E
SCHEMBL13409353 0.71 CYP3A4 (0.46) MAPTL3MBTL1TRPM8KDM4EALDH1A1
SCHEMBL16213745 0.69 LRRK2 (0.41) LRRK2MAOATRPM8KCNH2GAK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7705146-B2 Hepatitis C inhibitor peptide analogs BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-27 US disclosed