SCHEMBL8273373

SCHEMBL8273373

Bc1cc(C(=O)C(=O)c2ccc(OC)c(C)c2)ccc1C#N

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
ALOX15 P16050 1/20 0.43
RAB9A P51151 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
KDM4E B2RXH2 1/20 0.42
USP2 O75604 1/20 0.42
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
TAS1R3 Q7RTX0 5/20 0.41
TAS1R1 Q7RTX1 5/20 0.41
F11 P03951 1/20 0.39
CFTR P13569 1/20 0.39
IMPDH2 P12268 2/20 0.39
IMPDH1 P20839 1/20 0.39
HPGD P15428 1/20 0.39
POLB P06746 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3534758 0.83 ALDH1A1 (0.49) ALDH1A1ALOX15RAB9AMEN1KMT2A
SCHEMBL13082597 0.77 TSHR (0.63) ALDH1A1ALOX15RAB9AMEN1KMT2A
SCHEMBL15624016 0.76 CA1 (0.47) ALDH1A1ALOX15MEN1KMT2AKDM4E
SCHEMBL3538604 0.74 CTSD (0.58) ALDH1A1RAB9AMEN1KMT2AKDM4E
SCHEMBL13263912 0.74 ALDH1A1 (0.52) ALDH1A1RAB9AMEN1KMT2AKDM4E
SCHEMBL24890475 0.72 ALOX15 (0.51) ALDH1A1ALOX15RAB9ATAS1R3TAS1R1
SCHEMBL7621232 0.72 ALOX15 (0.51) ALDH1A1ALOX15RAB9ATAS1R3TAS1R1
SCHEMBL11577171 0.71 CYP1A2 (0.70) ALDH1A1ALOX15TAS1R3TAS1R1HPGD
SCHEMBL1419879 0.71 ALDH1A1 (0.62) ALDH1A1RAB9AKDM4EUSP2F11
SCHEMBL7001839 0.71 ALDH1A1 (0.65) ALDH1A1MEN1KMT2AKDM4EUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006009653-A1 AMINO-5,5-DIPHENYLIMIDAZOLONE DERIVATIVES FOR THE INHIBITION OF BETA-SECRETASE WYETH (US) 2006-01-26 WO disclosed