SCHEMBL8274131

SCHEMBL8274131

c1cc2c(ccc3occc32)cn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 2/20 0.45
IMPDH2 P12268 4/20 0.42
NFKB1 P19838 1/20 0.41
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
DYRK1A Q13627 1/20 0.41
KDM4E B2RXH2 2/20 0.40
LMNA P02545 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
MAPKAPK2 P49137 1/20 0.40
ERN1 O75460 1/20 0.39
HTR2A P28223 2/20 0.37
HTR2C P28335 2/20 0.37
HTT P42858 2/20 0.37
CDK4 P11802 1/20 0.37
CCND1 P24385 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2047737 0.85 DYRK1A (0.41) DRD1NFKB1MAOAMAOBDYRK1A
SCHEMBL31061858 0.81 DRD1 (0.39) DRD1IMPDH2NFKB1DYRK1AKDM4E
SCHEMBL445595 0.78 IMPDH2 (0.58) IMPDH2MAOAMAOBDYRK1AKDM4E
Bromide SCHEMBL27922950 0.76 IMPDH2 (0.56) IMPDH2MAOAMAOBDYRK1AKDM4E
Pyrazine SCHEMBL29129778 0.76 TDP1 (0.44) NFKB1MAOAMAOBDYRK1AKDM4E
SCHEMBL8274128 0.74 IMPDH2 (0.43) DRD1IMPDH2MAOAMAOBDYRK1A
SCHEMBL4429415 0.73 PAX8 (0.48) NFKB1MAOAMAOBDYRK1AKDM4E
Pyridine SCHEMBL28575847 0.73 HSD17B10 (0.41) NFKB1MAOAMAOBDYRK1AKDM4E
Pyrimidine SCHEMBL29096576 0.73 HSD17B10 (0.41) NFKB1MAOAMAOBDYRK1AKDM4E
SCHEMBL88833 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006000085-A1 HEPATITIS C INHIBITOR PEPTIDE ANALOGS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2006-01-05 WO disclosed