SCHEMBL8274136

SCHEMBL8274136

c1cc2c3c(ccc2cn1)CCO3

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 4/20 0.39
LMNA P02545 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
KDM4E B2RXH2 1/20 0.37
MAPKAPK2 P49137 1/20 0.37
ACHE P22303 1/20 0.36
ERN1 O75460 1/20 0.36
CDC7 O00311 1/20 0.35
CYP19A1 P11511 2/20 0.35
CYP11B1 P15538 2/20 0.35
CYP11B2 P19099 2/20 0.35
KDM4C Q9H3R0 1/20 0.34
HTT P42858 1/20 0.34
CDK4 P11802 1/20 0.34
CCND1 P24385 1/20 0.34
PARP1 P09874 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22065919 0.86 CLK1 (0.37) KDM4EACHEKDM4CHTTPARP1
SCHEMBL22744586 0.80 SSTR4 (0.51) IMPDH2CYP1A2CYP3A4CYP2C19KDM4E
SCHEMBL3968484 0.77 IDO1 (0.44) IMPDH2LMNACYP1A2CYP3A4CYP2D6
SCHEMBL8274137 0.72 IDO1 (0.40) IMPDH2LMNACYP1A2CYP3A4CYP2D6
SCHEMBL3971384 0.70 KDM4E (0.43) IMPDH2LMNACYP1A2CYP3A4CYP2D6
SCHEMBL445595 0.70 IMPDH2 (0.58) IMPDH2LMNACYP1A2CYP3A4CYP2D6
SCHEMBL22065129 0.69 IL5 (0.46) CYP1A2ACHEPARP1
SCHEMBL8276161 0.68 CYP2A6 (0.34) PARP1
SCHEMBL15665250 0.68 PARP1 (0.36) KDM4CPARP1
SCHEMBL1536439 0.68 LMNA (0.41) LMNACYP3A4PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006000085-A1 HEPATITIS C INHIBITOR PEPTIDE ANALOGS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2006-01-05 WO disclosed