SCHEMBL8276161

SCHEMBL8276161

Cc1nccc2c3c(ccc12)CCO3

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.34
PDE3B Q13370 2/20 0.33
PDE3A Q14432 2/20 0.33
PKM P14618 1/20 0.33
PARP1 P09874 1/20 0.33
EPHB4 P54760 1/20 0.32
BRD4 O60885 1/20 0.32
DAO P14920 1/20 0.31
NR3C1 P04150 1/20 0.31
PGR P06401 1/20 0.31
NR3C2 P08235 1/20 0.31
AR P10275 1/20 0.31
MAOA P21397 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15665250 0.80 PARP1 (0.36) PARP1DAO
SCHEMBL1536439 0.80 LMNA (0.41) PARP1DAO
SCHEMBL8277400 0.80 PDE3B (0.38) PDE3BPDE3APARP1
SCHEMBL8272974 0.80 PARP1 (0.30) PARP1
SCHEMBL7822600 0.80 ATM (0.35) PARP1
SCHEMBL8272975 0.78 ADRA2A (0.42) CYP2A6PDE3BPDE3APKMMAOA
SCHEMBL8271695 0.77 SMN1; SMN2 (0.36) PARP1
SCHEMBL13409371 0.76 LRRK2 (0.34)
SCHEMBL15178727 0.75 PDE10A (0.34) BRD4
SCHEMBL8277403 0.73 DRD1 (0.39) CYP2A6PDE3BPDE3APKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1771453-B1 HEPATITIS C INHIBITOR DIPEPTIDE ANALOGS BOEHRINGER INGELHEIM INT (DE) 2012-05-30 EP disclosed
WO-2006007700-A1 HEPATITIS C INHIBITOR DIPEPTIDE ANALOGS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2006-01-26 WO disclosed