SCHEMBL8277403

SCHEMBL8277403

Cc1nccc2c3c(ccc12)OCC3

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 5/20 0.39
EED O75530 8/20 0.37
PKM P14618 1/20 0.36
SUZ12 Q15022 2/20 0.34
EZH2 Q15910 2/20 0.34
CYP2A6 P11509 1/20 0.34
PDE3B Q13370 2/20 0.33
PDE3A Q14432 2/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
CHRM2 P08172 1/20 0.33
ADRA2A P08913 1/20 0.33
SLC18A2 Q05940 1/20 0.33
PDE4D Q08499 1/20 0.33
SLC9A1 P19634 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17190972 0.80 DRD1 (0.46) DRD1EEDPKMSUZ12EZH2
SCHEMBL1536445 0.80 LMNA (0.41) DRD1SLC9A1
SCHEMBL7818979 0.80 HTR2A (0.33) DRD1PKMSLC9A1
SCHEMBL8272973 0.80 HTR2A (0.35) DRD1EEDSUZ12EZH2ALDH1A1
SCHEMBL8271685 0.80 DRD1 (0.39) DRD1EEDSUZ12EZH2SLC9A1
SCHEMBL8276151 0.80 PDE3B (0.38) DRD1EEDSUZ12EZH2PDE3B
SCHEMBL8272975 0.78 ADRA2A (0.42) PKMCYP2A6PDE3BPDE3AALDH1A1
SCHEMBL13409369 0.76 DRD1 (0.37) DRD1EEDSUZ12EZH2
SCHEMBL8276161 0.73 CYP2A6 (0.34) PKMCYP2A6PDE3BPDE3A
SCHEMBL12266516 0.71 CYP2A6 (0.56) CYP2A6PDE3BPDE3AALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1771453-B1 HEPATITIS C INHIBITOR DIPEPTIDE ANALOGS BOEHRINGER INGELHEIM INT (DE) 2012-05-30 EP disclosed
WO-2006007700-A1 HEPATITIS C INHIBITOR DIPEPTIDE ANALOGS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2006-01-26 WO disclosed