SCHEMBL8280205

SCHEMBL8280205

CNCc1ccccc1-c1ccsc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.54
PRMT6 Q96LA8 1/20 0.51
CYP2A6 P11509 2/20 0.42
CYP2B6 P20813 2/20 0.42
CYP2E1 P05181 1/20 0.42
OPRL1 P41146 1/20 0.40
PTPRC P08575 1/20 0.38
ADORA1 P30542 1/20 0.38
BCHE P06276 1/20 0.37
IFNAR1 P17181 1/20 0.37
KIT P10721 1/20 0.37
FLT1 P17948 1/20 0.37
KDR P35968 1/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
EDNRA P25101 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
SLC6A2 P23975 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12819940 0.80 CYP2A6 (0.47) CYP2A6CYP2B6CYP2E1OPRL1PTPRC
SCHEMBL30340124 0.80 CYP2A6 (0.47) CYP2A6CYP2B6CYP2E1OPRL1PTPRC
SCHEMBL15525017 0.78 SLC6A2 (0.49) CYP2A6CYP2B6CYP2E1OPRL1PTPRC
SCHEMBL417693 0.77 LTA4H (0.55) LTA4HPRMT6CYP3A4SLC6A2SLC6A4
SCHEMBL28754758 0.77 CYP2A6 (0.48) PRMT6CYP2A6CYP2B6CYP2E1PTPRC
SCHEMBL22548895 0.77 CYP2A6 (0.44) PRMT6CYP2A6CYP2B6CYP2E1PTPRC
SCHEMBL21480391 0.77 CYP2A6 (0.47) CYP2A6CYP2B6CYP2E1PTPRCBCHE
SCHEMBL477489 0.77 CYP2A6 (0.47) CYP2A6CYP2B6CYP2E1PTPRCKIT
SCHEMBL7502553 0.77 CYP2A6 (0.47) CYP2A6CYP2B6CYP2E1PTPRCBCHE
SCHEMBL3181212 0.77 CYP2A6 (0.47) CYP2A6CYP2B6CYP2E1PTPRCBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005090354-A1 PYRAZOLO[3,4-b] PYRIDINE COMPOUNDS, AND THEIR USE AS PDE4 INHIBITORS GLAXO GROUP LIMITED (GB) 2005-09-29 WO disclosed