SCHEMBL8282113

SCHEMBL8282113

CCOc1ccc(-c2nnc(C)n2-c2ccc(C)cc2)cc1C

nearest known ligand 0.71

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
OXTR P30559 9/20 0.71
AVPR1A P37288 7/20 0.54
AVPR2 P30518 3/20 0.51
HPGD P15428 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CACNA2D1 P54289 1/20 0.43
BRD4 O60885 3/20 0.41
MAPT P10636 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
UCHL3 P15374 1/20 0.40
GRK6 P43250 1/20 0.40
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8279809 0.90 OXTR (0.68) OXTRAVPR1AAVPR2HPGDSMN1; SMN2
SCHEMBL8281669 0.86 OXTR (0.77) OXTRAVPR1AAVPR2HPGDSMN1; SMN2
SCHEMBL8282112 0.83 OXTR (1.00) OXTRAVPR1AAVPR2
SCHEMBL8282111 0.82 OXTR (0.61) OXTRAVPR1AAVPR2HPGDSMN1; SMN2
SCHEMBL8280928 0.79 OXTR (0.58) OXTRAVPR1AAVPR2HPGDSMN1; SMN2
SCHEMBL8281723 0.79 OXTR (0.58) OXTRAVPR1AAVPR2MAPTNPSR1
SCHEMBL6511017 0.72 OXTR (0.80) OXTRAVPR1AAVPR2
SCHEMBL27530845 0.70 SMN1; SMN2 (0.79) OXTRAVPR1AAVPR2HPGDSMN1; SMN2
SCHEMBL8282084 0.70 OXTR (0.81) OXTRAVPR1AAVPR2
SCHEMBL8281027 0.69 OXTR (1.00) OXTRAVPR1AAVPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005082866-A2 SUBSTITUTED 1, 2, 4- TRIAZOLE DERIVATIVES AS OXYTOCIN ANTAGONISTS PFIZER LIMITED (GB) 2005-09-09 WO disclosed