SCHEMBL8282943

SCHEMBL8282943

CN(C(=O)CCCCC(c1ccc(F)cc1)c1ccc(F)cc1)[C@@H]1CCN(Cc2ccccc2)C1

nearest known ligand 0.58

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 17/20 0.58
KCNH2 Q12809 1/20 0.48
MCHR1 Q99705 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13920772 0.80 CCR5 (0.61) CCR5KCNH2
SCHEMBL4461059 0.76 CCR5 (0.44) CCR5KCNH2
SCHEMBL1220330 0.76 OPRM1 (0.59) KCNH2
SCHEMBL3817982 0.76 OPRM1 (0.59) KCNH2
SCHEMBL6703964 0.76 KCNH2 (0.79) CCR5KCNH2
SCHEMBL4474101 0.75 KCNH2 (0.58) CCR5KCNH2
SCHEMBL4466197 0.75 KCNH2 (0.58) CCR5KCNH2
Hydrochloric Acid SCHEMBL4469376 0.75 OPRM1 (0.57) KCNH2
SCHEMBL10654998 0.75 LTA4H (0.64) KCNH2
Hydrochloric Acid SCHEMBL4469375 0.75 OPRM1 (0.57) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7507760-B2 N-type calcium channel blockers NEUROMED PHARMACEUTICALS LTD. (CA) 2009-03-24 US disclosed
US-7507760-B2 N-type calcium channel blockers NEUROMED PHARMACEUTICALS LTD. (CA) 2009-03-24 US disclosed
WO-2005070919-A1 N-TYPE CALCIUM CHANNEL BLOCKERS NEUROMED PHARMACEUTICALS LTD. (CA) 2005-08-04 WO disclosed