SCHEMBL8285202

SCHEMBL8285202

COCCNc1cc(C)nc2c1c(=O)cc(Nc1ccccc1)n2-c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 2/20 0.47
PDE11A Q9HCR9 1/20 0.42
KCNH3 Q9ULD8 4/20 0.42
CFTR P13569 1/20 0.38
KDM4E B2RXH2 5/20 0.38
MAPK1 P28482 3/20 0.38
HSD17B10 Q99714 2/20 0.38
GAA P10253 4/20 0.38
HPGD P15428 4/20 0.38
ALDH1A1 P00352 4/20 0.38
ATM Q13315 2/20 0.38
GLA P06280 2/20 0.38
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38
NPSR1 Q6W5P4 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
POLB P06746 2/20 0.35
LMNA P02545 2/20 0.35
MAPT P10636 1/20 0.35
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8285238 0.85 PDE11A (0.49) PDE11AKDM4EMAPK1GAAHPGD
SCHEMBL8285244 0.84 PDE11A (0.44) PDE11AKDM4EMAPK1GAAHPGD
SCHEMBL8287830 0.83 PDE11A (0.48) PDE11AKDM4EMAPK1GAAHPGD
SCHEMBL8286379 0.83 PDE11A (0.43) PDE11AKDM4EMAPK1GAAHPGD
SCHEMBL8286423 0.82 KCNH3 (0.42) NCF1PDE11AKCNH3CFTRKDM4E
SCHEMBL8361761 0.82 ALDH1A1 (0.42) PDE11AKDM4EMAPK1HSD17B10GAA
SCHEMBL8287405 0.82 OPRK1 (0.53) PDE11AKDM4EMAPK1GAAHPGD
SCHEMBL8287832 0.80 PDE11A (0.47) PDE11AKDM4EMAPK1GAAHPGD
SCHEMBL8361762 0.80 OPRK1 (0.41) PDE11AKDM4EMAPK1HSD17B10GAA
SCHEMBL8286452 0.80 PDE11A (0.44) PDE11AKDM4EGAAHPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005091857-A2 1,6-NAPHTHYRIDINE AND 1,8-NAPHTHYRIDINE DERIVATIVES AND THEIR USE TO TREAT DIABETES AND RELATED DISORDERS BAYER PHARMACEUTICALS CORPORATION (US) 2005-10-06 WO disclosed
WO-2003027112-A1 1, 8-NAPHTHYRIDINE DERIVATIVES AS ANTIDIABETICS BAYER PHARMACEUTICALS CORPORATION (US) 2003-04-03 WO disclosed