SCHEMBL8286102

SCHEMBL8286102

CCC(NC)c1ccccc1C

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.43
ACP3 P15309 1/20 0.38
TSHR P16473 2/20 0.36
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 2/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
SLC6A3 Q01959 1/20 0.36
KCNH2 Q12809 1/20 0.36
CTSA P10619 8/20 0.36
ACHE P22303 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13076103 0.84 ESR1 (0.41) ESR1ACP3TSHRSLC6A2SLC6A4
SCHEMBL8284261 0.84 ADRA2A (0.37) ESR1TSHRSLC6A2CYP3A4CYP2D6
SCHEMBL11628582 0.82 ESR1 (0.42) ESR1ACP3TSHRSLC6A2SLC6A4
SCHEMBL24222490 0.81 ADRB1 (0.36) ESR1CYP2D6CTSA
SCHEMBL8995496 0.81 ESR1 (0.38) ESR1ACP3SLC6A2SLC6A4CYP3A4
SCHEMBL24129481 0.81 ALDH1A1 (0.45) TSHRSLC6A2CYP3A4CYP2D6ACHE
SCHEMBL3956324 0.79 SCN1A (0.43) ESR1ACP3TSHRCTSA
SCHEMBL11128128 0.79 TDP1 (0.42) ESR1ACP3TSHRCYP3A4CTSA
SCHEMBL13075570 0.78 TAAR1 (0.37) SLC6A2SLC6A4CYP3A4CYP2D6SLC6A3
SCHEMBL8284300 0.78 CYP3A4 (0.39) TSHRSLC6A2SLC6A4CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022139228-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE COMPRISING SAME, MANUFACTURING METHOD THEREFOR, AND COMPOSITION FOR ORGANIC MATERIAL LAYER 엘티소재주식회사 2022-06-30 WO disclosed
US-20070111995-A1 Pyrazolo [3,4-B] pyridine Compounds and Their Use as Phosphodiesterase Inhibitors GLAXO GROUP LIMITED (GB) 2007-05-17 US disclosed
WO-2005058892-A1 PYRAZOLO [3,4-B] PYRIDINE COMPOUNDS, AND THEIR USE AS PHOSPHODIESTERASE INHIBITORS GLAXO GROUP LIMITED (GB) 2005-06-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070111995-A1 Pyrazolo [3,4-B] pyridine Compounds and Their Use as Phosphodiesterase Inhibitors PDE4B, PDE3B, PDE4A ESR1 4063/4885ACP3 338/4885TSHR 1576/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.