SCHEMBL8287708

SCHEMBL8287708

Cc1c(N)cccc1C(=O)NCC(=O)N1CCC[C@H]1C=O

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PREP P48147 18/20 0.47
FAP Q12884 5/20 0.47
DPP8 Q6V1X1 1/20 0.47
DPP9 Q86TI2 1/20 0.47
DPP7 Q9UHL4 1/20 0.42
DPP4 P27487 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12031852 0.87 PREP (0.47) PREPFAPDPP8DPP9DPP7
SCHEMBL8286743 0.85 PREP (0.50) PREPFAPDPP8DPP9
SCHEMBL8288913 0.84 PREP (0.50) PREPFAPDPP8DPP9DPP4
SCHEMBL8286887 0.84 FAP (0.47) PREPFAPDPP8DPP9
SCHEMBL8287698 0.83 PREP (0.47) PREPFAPDPP8DPP9DPP7
SCHEMBL12031643 0.81 PREP (0.51) PREPFAPDPP8DPP9DPP7
SCHEMBL12031716 0.80 PREP (0.47) PREPFAPDPP8DPP9DPP7
SCHEMBL8288851 0.80 PREP (0.52) PREPFAPDPP8DPP9DPP7
SCHEMBL16281614 0.80 PREP (0.60) PREPFAPDPP4
SCHEMBL12949922 0.80 PREP (0.54) PREPFAPDPP8DPP9DPP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2399915-A1 Process and intermediates for the preparation of aspartic acetal caspase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-12-28 EP disclosed
WO-2005085236-A2 CASPASE INHIBITORS AND USES THEREOF VERTEX PHARMACEUTICALS INCORPORATED (US) 2005-09-15 WO disclosed