SCHEMBL8288403

SCHEMBL8288403

CNC(=O)C(CCC1CCCCC1)CC1CCCCC1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
KMT2A Q03164 1/20 0.43
LTA4H P09960 1/20 0.43
MMP1 P03956 7/20 0.42
MMP13 P45452 3/20 0.42
METAP1 P53582 2/20 0.40
CTSK P43235 2/20 0.39
METAP2 P50579 2/20 0.39
CTSS P25774 1/20 0.39
HPGD P15428 1/20 0.38
MMP3 P08254 1/20 0.38
SIGMAR1 Q99720 1/20 0.37
CTSL P07711 1/20 0.37
CTSB P07858 1/20 0.37
CTSH P09668 1/20 0.37
CPB2 Q96IY4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13500299 0.98 ALDH1A1 (0.41) ALDH1A1KMT2ALTA4HMMP1MMP13
SCHEMBL13500292 0.97 ALDH1A1 (0.40) ALDH1A1KMT2ALTA4HMMP1MMP13
SCHEMBL13500291 0.97 MMP1 (0.42) ALDH1A1KMT2ALTA4HMMP1MMP13
SCHEMBL13500158 0.97 ALDH1A1 (0.40) ALDH1A1KMT2ALTA4HMMP1MMP13
SCHEMBL13501752 0.93 MMP1 (0.39) ALDH1A1KMT2ALTA4HMMP1MMP13
SCHEMBL13500153 0.91 MMP1 (0.37) ALDH1A1KMT2ALTA4HMMP1MMP13
SCHEMBL9456 0.87 ALDH1A1 (0.49) ALDH1A1KMT2ALTA4HMMP1MMP13
SCHEMBL13725530 0.86 MMP1 (0.39) ALDH1A1KMT2ALTA4HMMP1MMP13
SCHEMBL13500182 0.85 ALDH1A1 (0.47) ALDH1A1KMT2ALTA4HMMP1MMP13
SCHEMBL13500293 0.84 MMP1 (0.37) ALDH1A1KMT2ALTA4HMMP1MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2335701-A1 Heterocyclic aspartyl protease inhibitors Schering Corporation (US) 2011-06-22 EP disclosed
EP-2153832-A2 Heterocyclic aspartyl protease inhibitors SCHERING CORPORATION (US) 2010-02-17 EP disclosed
EP-1838304-B1 HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS SCHERING CORP (US) 2009-08-19 EP disclosed
WO-2005058311-A1 HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS SCHERING CORPORATION (US) 2005-06-30 WO disclosed