SCHEMBL8288554

SCHEMBL8288554

CC1CCc2c(sc(NC(=O)c3ccccc3C(=O)O)c2N)C1

nearest known ligand 0.72

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.72
RAB9A P51151 2/20 0.72
ALDH1A1 P00352 2/20 0.72
L3MBTL1 Q9Y468 2/20 0.72
TP53 P04637 3/20 0.59
PDE4B Q07343 2/20 0.56
PDE4D Q08499 2/20 0.56
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
TNF P01375 2/20 0.53
NOD1 Q9Y239 2/20 0.53
MAPT P10636 6/20 0.52
NPSR1 Q6W5P4 1/20 0.52
SAE1 Q9UBE0 1/20 0.52
UBA2 Q9UBT2 1/20 0.52
RORC P51449 1/20 0.52
ALOX12 P18054 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21247231 0.81 MAPT (0.76) NPC1RAB9AALDH1A1L3MBTL1TP53
SCHEMBL8288708 0.81 TP53 (0.67) NPC1RAB9AALDH1A1L3MBTL1TP53
SCHEMBL2182372 0.74 TP53 (0.80) NPC1RAB9AALDH1A1L3MBTL1TP53
SCHEMBL15281365 0.73 CCR6 (0.56) NPC1RAB9AALDH1A1L3MBTL1TP53
SCHEMBL21247383 0.69 MAPT (0.73) NPC1RAB9AALDH1A1L3MBTL1TP53
SCHEMBL21346818 0.69 FLT3 (0.70) NPC1RAB9AALDH1A1L3MBTL1TP53
SCHEMBL13744456 0.68 NPC1 (0.74) NPC1RAB9AL3MBTL1TP53MEN1
SCHEMBL23850645 0.68 RORC (1.00) NPC1RAB9AALDH1A1L3MBTL1TP53
SCHEMBL918283 0.68 MAPT (1.00) NPC1RAB9AALDH1A1L3MBTL1TP53
SCHEMBL8288764 0.68 FLT3 (0.78) NPC1RAB9AALDH1A1L3MBTL1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005033102-A2 THIOPHENE-BASED COMPOUNDS EXHIBITING ATP-UTILIZING ENZYME INHIBITORY ACTIVITY, AND COMPOSITIONS, AND USES THEREOF AMPHORA DISCOVERY CORPORATION (US) 2005-04-14 WO disclosed