SCHEMBL8288708

SCHEMBL8288708

Nc1c(NC(=O)c2ccccc2C(=O)O)sc2c1CCCC2

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.67
KMT2A Q03164 6/20 0.61
MEN1 O00255 5/20 0.61
FLT3 P36888 2/20 0.60
TNF P01375 1/20 0.60
NOD1 Q9Y239 1/20 0.60
FABP4 P15090 1/20 0.59
FABP5 Q01469 1/20 0.59
RAB9A P51151 6/20 0.59
NPC1 O15118 5/20 0.59
MAPT P10636 4/20 0.59
LMNA P02545 2/20 0.59
SMN1; SMN2 Q16637 2/20 0.59
L3MBTL1 Q9Y468 1/20 0.57
CFTR P13569 1/20 0.56
ALDH1A1 P00352 2/20 0.55
HPGD P15428 2/20 0.55
POLB P06746 1/20 0.53
ESR2 Q92731 1/20 0.53
CTDSP1 Q9GZU7 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13744456 0.86 NPC1 (0.74) TP53KMT2AMEN1FLT3TNF
SCHEMBL8288764 0.85 FLT3 (0.78) TP53KMT2AMEN1FLT3TNF
SCHEMBL15281390 0.81 MAPK10 (0.77) TP53KMT2AMEN1RAB9ANPC1
SCHEMBL8288554 0.81 NPC1 (0.72) TP53KMT2AMEN1TNFNOD1
SCHEMBL23493865 0.81 TP53 (1.00) TP53KMT2AMEN1FLT3TNF
SCHEMBL21247391 0.79 MEN1 (0.95) TP53KMT2AMEN1FLT3TNF
SCHEMBL20339108 0.78 L3MBTL1 (0.67) TP53KMT2AMEN1TNFNOD1
SCHEMBL8290453 0.77 LMNA (0.64) KMT2AMEN1MAPTLMNAALDH1A1
SCHEMBL21247135 0.76 MEN1 (1.00) TP53KMT2AMEN1FLT3TNF
SCHEMBL23928917 0.75 MEN1 (1.00) TP53KMT2AMEN1TNFNOD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005033102-A2 THIOPHENE-BASED COMPOUNDS EXHIBITING ATP-UTILIZING ENZYME INHIBITORY ACTIVITY, AND COMPOSITIONS, AND USES THEREOF AMPHORA DISCOVERY CORPORATION (US) 2005-04-14 WO disclosed