SCHEMBL8288690

SCHEMBL8288690

CC(C)NC(=O)Nc1sc2c(c1C(N)=O)C(C)CCC2

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 2/20 0.58
PDE4D Q08499 2/20 0.58
ABCC1 P33527 1/20 0.49
ABCG2 Q9UNQ0 1/20 0.49
CXCR2 P25025 10/20 0.48
CXCR4 P61073 4/20 0.48
KIF11 P52732 1/20 0.45
FLT3 P36888 3/20 0.43
KDM4E B2RXH2 2/20 0.43
MAPK1 P28482 1/20 0.43
MEN1 O00255 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C19 P33261 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8288836 0.84 PDE4B (0.57) PDE4BPDE4DABCC1ABCG2CXCR2
SCHEMBL3913969 0.82 FLT3 (0.64) PDE4BPDE4DABCC1ABCG2CXCR2
SCHEMBL8289710 0.78 KDM4E (0.70) FLT3KDM4EMAPK1MEN1CYP1A2
SCHEMBL5459748 0.78 FLT3 (0.70) FLT3KDM4EMAPK1MEN1CYP1A2
SCHEMBL8289722 0.78 PDE4B (0.52) PDE4BPDE4DABCC1ABCG2CXCR2
SCHEMBL5462746 0.77 MAPT (0.69) PDE4BPDE4DKDM4E
SCHEMBL8290436 0.77 FLT3 (0.68) FLT3KDM4EMAPK1MEN1CYP1A2
SCHEMBL5453397 0.75 PTPN1 (0.53) PDE4BPDE4DFLT3KDM4EMEN1
SCHEMBL8290782 0.74 ALDH1A1 (0.53) PDE4BPDE4DABCC1ABCG2CXCR2
SCHEMBL8290431 0.72 ANO1 (0.72) PDE4BPDE4DKDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005033102-A2 THIOPHENE-BASED COMPOUNDS EXHIBITING ATP-UTILIZING ENZYME INHIBITORY ACTIVITY, AND COMPOSITIONS, AND USES THEREOF AMPHORA DISCOVERY CORPORATION (US) 2005-04-14 WO disclosed