SCHEMBL8290782

SCHEMBL8290782

CC1CCCc2sc(N)c(C(N)=O)c21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.53
MAPT P10636 11/20 0.53
KDM4E B2RXH2 9/20 0.53
HPGD P15428 8/20 0.53
HSD17B10 Q99714 6/20 0.53
MEN1 O00255 5/20 0.53
KMT2A Q03164 5/20 0.53
USP2 O75604 1/20 0.53
RECQL P46063 1/20 0.53
ALOX15 P16050 6/20 0.52
MAPK1 P28482 2/20 0.51
PDE4B Q07343 1/20 0.47
PDE4D Q08499 1/20 0.47
LMNA P02545 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
ANO1 Q5XXA6 1/20 0.46
ABCC1 P33527 1/20 0.43
ABCG2 Q9UNQ0 1/20 0.43
CXCR2 P25025 5/20 0.43
LIMK1 P53667 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3911820 0.80 GAA (0.61) ALDH1A1MAPTKDM4EHPGDHSD17B10
SCHEMBL3913969 0.76 FLT3 (0.64) ALDH1A1MAPTKDM4EHPGDHSD17B10
SCHEMBL8289722 0.76 PDE4B (0.52) ALDH1A1MAPTKDM4EHSD17B10MEN1
SCHEMBL22543334 0.76 LIMK1 (0.39) ALDH1A1MAPTKDM4EHPGDHSD17B10
SCHEMBL8288690 0.74 PDE4B (0.58) KDM4EMEN1KMT2AMAPK1PDE4B
SCHEMBL8288836 0.74 PDE4B (0.57) KDM4EMEN1KMT2AMAPK1PDE4B
SCHEMBL22543319 0.73 ABCC1 (0.38) ALDH1A1MAPTKDM4EHPGDHSD17B10
SCHEMBL14829495 0.72 ALDH1A1 (0.44) ALDH1A1MAPTKDM4EHPGDHSD17B10
SCHEMBL21603773 0.71 ALDH1A1 (0.61) ALDH1A1MAPTKDM4EHPGDHSD17B10
SCHEMBL5449503 0.70 ALDH1A1 (0.47) ALDH1A1MAPTKDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005033102-A2 THIOPHENE-BASED COMPOUNDS EXHIBITING ATP-UTILIZING ENZYME INHIBITORY ACTIVITY, AND COMPOSITIONS, AND USES THEREOF AMPHORA DISCOVERY CORPORATION (US) 2005-04-14 WO disclosed