SCHEMBL8290409

SCHEMBL8290409

NC(=O)c1c(NC(=O)c2ccc(C(F)(F)F)cc2F)sc2c1CCCC2

nearest known ligand 0.70

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 9/20 0.70
RAB9A P51151 9/20 0.70
FLT3 P36888 9/20 0.61
CFTR P13569 1/20 0.58
MAPT P10636 3/20 0.57
SMN1; SMN2 Q16637 3/20 0.57
ALDH1A1 P00352 2/20 0.57
KMT2A Q03164 3/20 0.56
MEN1 O00255 2/20 0.56
CASP3 P42574 1/20 0.56
SENP7 Q9BQF6 1/20 0.56
POLB P06746 1/20 0.56
XPO1 O14980 1/20 0.56
LMNA P02545 2/20 0.55
KDM4E B2RXH2 1/20 0.55
ALOX15 P16050 1/20 0.55
TSHR P16473 1/20 0.55
HSD17B10 Q99714 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8288680 0.98 NPC1 (0.67) NPC1RAB9AFLT3CFTRMAPT
SCHEMBL8289498 0.85 FLT3 (0.79) NPC1RAB9AFLT3MAPTSMN1; SMN2
SCHEMBL8288685 0.84 FLT3 (0.77) NPC1RAB9AFLT3MAPTSMN1; SMN2
SCHEMBL8289720 0.83 NPC1 (0.73) NPC1RAB9AFLT3CFTRMAPT
SCHEMBL12218351 0.81 NPC1 (0.98) NPC1RAB9AFLT3CFTRMAPT
SCHEMBL8290644 0.79 NPC1 (0.96) NPC1RAB9AFLT3CFTRMAPT
SCHEMBL5453475 0.78 ANO1 (0.65) NPC1RAB9AFLT3MAPTSMN1; SMN2
SCHEMBL8290852 0.78 FLT3 (0.75) NPC1RAB9AFLT3MAPTSMN1; SMN2
SCHEMBL8289579 0.78 NPC1 (0.78) NPC1RAB9AFLT3CFTRMAPT
SCHEMBL8289526 0.78 RAB9A (0.95) NPC1RAB9AFLT3MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005033102-A2 THIOPHENE-BASED COMPOUNDS EXHIBITING ATP-UTILIZING ENZYME INHIBITORY ACTIVITY, AND COMPOSITIONS, AND USES THEREOF AMPHORA DISCOVERY CORPORATION (US) 2005-04-14 WO disclosed