SCHEMBL8290727

SCHEMBL8290727

Cc1sc(NC(=O)c2ccc3c(c2)OCO3)c(C(N)=O)c1C

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 8/20 0.70
RAB9A P51151 8/20 0.70
FLT3 P36888 2/20 0.65
ALDH1A1 P00352 4/20 0.64
HPGD P15428 3/20 0.64
KDM4E B2RXH2 2/20 0.64
LMNA P02545 1/20 0.64
MAPT P10636 5/20 0.61
GAA P10253 2/20 0.61
MEN1 O00255 2/20 0.61
KMT2A Q03164 2/20 0.61
POLB P06746 1/20 0.61
GRIN2C Q14957 1/20 0.60
SMN1; SMN2 Q16637 3/20 0.57
CASP3 P42574 2/20 0.57
SENP7 Q9BQF6 2/20 0.57
PKM P14618 1/20 0.52
NFKB1 P19838 1/20 0.52
NFKB2 Q00653 1/20 0.52
RELA Q04206 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13799001 0.87 NPC1 (0.60) NPC1RAB9AALDH1A1HPGDMAPT
SCHEMBL7676531 0.81 MAPK8 (0.63) NPC1RAB9AALDH1A1HPGDKDM4E
SCHEMBL7003572 0.79 MAPT (0.80) NPC1RAB9AALDH1A1HPGDKDM4E
SCHEMBL7669932 0.79 MAPT (0.80) NPC1RAB9AALDH1A1HPGDKDM4E
SCHEMBL22789369 0.79 FLT3 (1.00) NPC1RAB9AFLT3ALDH1A1HPGD
SCHEMBL7004549 0.78 FLT3 (0.68) NPC1RAB9AFLT3ALDH1A1HPGD
SCHEMBL7002672 0.77 FLT3 (1.00) NPC1RAB9AFLT3ALDH1A1HPGD
SCHEMBL7902809 0.75 GRIN2C (1.00) NPC1RAB9AFLT3ALDH1A1HPGD
SCHEMBL7003132 0.75 ALDH1A1 (0.64) NPC1RAB9AFLT3ALDH1A1HPGD
SCHEMBL5245843 0.74 MAPT (0.54) NPC1RAB9AFLT3ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005033102-A2 THIOPHENE-BASED COMPOUNDS EXHIBITING ATP-UTILIZING ENZYME INHIBITORY ACTIVITY, AND COMPOSITIONS, AND USES THEREOF AMPHORA DISCOVERY CORPORATION (US) 2005-04-14 WO disclosed