SCHEMBL8294356

SCHEMBL8294356

N[C@@H](CCCCNC(=O)c1coc(-c2ccccc2)n1)C(=O)N1CCC(F)(F)C1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.41
HDAC8 Q9BY41 2/20 0.41
HDAC6 Q9UBN7 2/20 0.41
TLR9 Q9NR96 5/20 0.39
TLR8 Q9NR97 5/20 0.39
TLR7 Q9NYK1 5/20 0.39
TBXAS1 P24557 3/20 0.39
DPP7 Q9UHL4 6/20 0.38
DPP4 P27487 3/20 0.38
KCNH2 Q12809 1/20 0.38
DPP8 Q6V1X1 4/20 0.38
ALDH1A1 P00352 1/20 0.38
PREP P48147 1/20 0.38
FAP Q12884 1/20 0.38
TGM2 P21980 1/20 0.38
DPP9 Q86TI2 3/20 0.38
ACKR3 P25106 1/20 0.37
TBXA2R P21731 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8293676 0.93 HDAC1 (0.44) HDAC1HDAC8HDAC6TLR9TLR8
SCHEMBL8294919 0.85 HDAC1 (0.45) HDAC1HDAC8HDAC6TLR9TLR8
SCHEMBL8293659 0.83 L3MBTL1 (0.40) DPP7DPP4KCNH2DPP8ALDH1A1
Hydrochloric Acid SCHEMBL6532979 0.81 DGAT1 (0.46)
Hydrochloric Acid SCHEMBL6532983 0.81 DGAT1 (0.46)
SCHEMBL8294350 0.79 ADAMTS7 (0.43) HDAC1HDAC6DPP7DPP4KCNH2
Hydrochloric Acid SCHEMBL6809246 0.79 HDAC3 (0.47) HDAC1
Hydrochloric Acid SCHEMBL6809256 0.77 DPP7 (0.38) DPP7DPP4KCNH2DPP8TGM2
SCHEMBL8293660 0.76 GAA (0.42) DPP7DPP4DPP8ALDH1A1DPP9
SCHEMBL8292700 0.75 HDAC1 (0.42) HDAC1DPP7DPP4KCNH2DPP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005019168-A2 FLUORINATED LYSINE DERIVATIVES AS DIPEPTIDYL PEPTIDASE IV INHIBITORS PFIZER PRODUCTS INC. (US) 2005-03-03 WO disclosed