SCHEMBL8294435

SCHEMBL8294435

CC(C)(C)OC(=O)N[C@@H](CC(=O)N1Cc2ccncc2CC1C(=O)NC1CC1)Cc1ccccc1F

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 13/20 0.41
TDP1 Q9NUW8 1/20 0.41
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
DRD2 P14416 2/20 0.37
CXCR3 P49682 2/20 0.36
SCN10A Q9Y5Y9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6249845 1.00 SCN9A (0.41) SCN9ATDP1CTSSCTSKDRD2
SCHEMBL8294434 0.97 SCN9A (0.41) SCN9ATDP1CTSSCTSKDRD2
SCHEMBL8293705 0.90 CTSS (0.42) SCN9ATDP1CTSSCTSKCXCR3
SCHEMBL8293704 0.89 KLK5 (0.42) SCN9ATDP1CTSSCTSKCXCR3
SCHEMBL8293702 0.87 CTSS (0.42) SCN9ATDP1CTSSCTSKCXCR3
SCHEMBL8293703 0.86 KLK5 (0.42) SCN9ATDP1CTSSCTSKCXCR3
SCHEMBL8293140 0.84 DPP4 (0.49)
SCHEMBL8294728 0.81 TDP1 (0.48) SCN9ATDP1CTSSCTSKCXCR3
SCHEMBL6253225 0.81 TDP1 (0.48) SCN9ATDP1CTSSCTSKCXCR3
SCHEMBL8293158 0.81 DPP4 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005056013-A1 DPP-IV INHIBITORS SANTHERA PHARMACEUTICALS (SCHWEIZ) GMBH (CH) 2005-06-23 WO disclosed