SCHEMBL8295708

SCHEMBL8295708

CC(C)C(NC(=O)OC(C)(C)C)c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.53
CTSS P25774 2/20 0.53
HDAC1 Q13547 1/20 0.51
ALDH1A1 P00352 2/20 0.50
GABRB1 P18505 1/20 0.47
GABRB2 P47870 1/20 0.47
MAPT P10636 1/20 0.47
ATM Q13315 1/20 0.47
POLB P06746 1/20 0.47
KMT2A Q03164 1/20 0.46
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA7 P43166 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12993554 1.00 CTSK (0.53) CTSKCTSSHDAC1ALDH1A1GABRB1
SCHEMBL13211538 0.89 CTSK (0.52) CTSKCTSSGABRB1GABRB2MAPT
SCHEMBL16622532 0.89 CTSK (0.52) CTSKCTSSGABRB1GABRB2MAPT
SCHEMBL4731613 0.89 CTSK (0.52) CTSKCTSSGABRB1GABRB2MAPT
SCHEMBL1908632 0.89 CTSK (0.52) CTSKCTSSGABRB1GABRB2MAPT
SCHEMBL16247215 0.88 CTSK (0.51) CTSKCTSSGABRB1GABRB2MAPT
SCHEMBL29839237 0.88 CTSK (0.51) CTSKCTSSGABRB1GABRB2MAPT
SCHEMBL15165758 0.88 KEAP1 (0.51) CTSKCTSSGABRB1GABRB2MAPT
SCHEMBL1573516 0.88 KEAP1 (0.51) CTSKCTSSGABRB1GABRB2MAPT
SCHEMBL5862225 0.88 KEAP1 (0.51) CTSKCTSSGABRB1GABRB2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7449447-B2 Peptidomimetic NS3-serine protease inhibitors of hepatitis C virus SCHERING CORPORATION (US) 2008-11-11 US disclosed
WO-2005021584-A2 NOVEL PEPTIDOMIMETIC NS3-SERINE PROTEASE INHIBITORS OF HEPATITIS C VIRUS SCHERING CORPORATION (US) 2005-03-10 WO disclosed