SCHEMBL5862225

SCHEMBL5862225

CC(C(=O)O)[C@@H](NC(=O)OC(C)(C)C)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 5/20 0.51
NFE2L2 Q16236 5/20 0.51
CTSK P43235 3/20 0.51
CTSS P25774 1/20 0.51
GABRB1 P18505 1/20 0.45
GABRB2 P47870 1/20 0.45
MAPT P10636 1/20 0.45
PPARA Q07869 2/20 0.45
PPARG P37231 1/20 0.45
ATM Q13315 1/20 0.45
ACE P12821 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15165758 1.00 KEAP1 (0.51) KEAP1NFE2L2CTSKCTSSGABRB1
SCHEMBL1573516 1.00 KEAP1 (0.51) KEAP1NFE2L2CTSKCTSSGABRB1
SCHEMBL13079942 0.90 CTSK (0.50) KEAP1NFE2L2CTSKCTSSGABRB1
SCHEMBL26647713 0.88 CTSS (0.47) KEAP1NFE2L2CTSKCTSSMAPT
SCHEMBL8295708 0.88 CTSK (0.53) CTSKCTSSGABRB1GABRB2MAPT
SCHEMBL12993554 0.88 CTSK (0.53) CTSKCTSSGABRB1GABRB2MAPT
SCHEMBL23205818 0.87 PPARG (0.47) KEAP1NFE2L2CTSKCTSSMAPT
SCHEMBL5862822 0.87 PPARG (0.47) KEAP1NFE2L2CTSKCTSSMAPT
SCHEMBL20521905 0.87 PPARG (0.47) KEAP1NFE2L2CTSKCTSSMAPT
SCHEMBL6513379 0.87 KEAP1 (0.42) KEAP1NFE2L2CTSKCTSSPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7041667-B1 CCR5 modulators PFIZER, INC. (US) 2006-05-09 US disclosed