SCHEMBL8296155

SCHEMBL8296155

OC1(c2ccccc2)CCN(CCC2(c3ccc(Cl)c(Cl)c3)CCCNC2)CC1

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 6/20 0.60
SLC6A4 P31645 6/20 0.60
SLC6A3 Q01959 4/20 0.60
TACR1 P25103 7/20 0.58
CYP2D6 P10635 2/20 0.56
TACR2 P21452 6/20 0.47
DRD2 P14416 2/20 0.45
DRD4 P21917 2/20 0.45
DRD3 P35462 2/20 0.45
TACR3 P29371 2/20 0.45
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
OPRM1 P35372 2/20 0.43
OPRL1 P41146 1/20 0.43
CCR5 P51681 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzaldehyde SCHEMBL6693667 0.86 SLC6A2 (0.49) SLC6A2SLC6A4SLC6A3TACR1CYP2D6
SCHEMBL3466336 0.82 SLC6A2 (0.63) SLC6A2SLC6A4SLC6A3TACR1CYP2D6
SCHEMBL3466330 0.82 SLC6A2 (0.63) SLC6A2SLC6A4SLC6A3TACR1CYP2D6
SCHEMBL8300496 0.81 SLC6A2 (0.54) SLC6A2SLC6A4SLC6A3TACR1CYP2D6
SCHEMBL7841995 0.81 TACR2 (0.58) TACR1TACR2TACR3
SCHEMBL7841999 0.81 TACR2 (0.58) TACR1TACR2TACR3
Hydrochloric Acid SCHEMBL8742517 0.81 SLC6A2 (0.53) SLC6A2SLC6A4SLC6A3TACR1CYP2D6
SCHEMBL8298555 0.80 TACR1 (0.75) TACR1TACR2TACR3OPRL1CCR5
Hydrochloric Acid SCHEMBL8742480 0.79 TACR1 (0.74) TACR1TACR2TACR3OPRL1
SCHEMBL7010561 0.79 TACR2 (0.61) SLC6A2SLC6A4SLC6A3TACR1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0512901-B1 Aminated polycyclic compounds and their enantiomers, process for their preparation and pharmaceutical compositions containing them SANOFI SA (FR) 1999-06-23 EP disclosed
US-5625060-A Polycyclic amine compounds and their enantiomers, their method of preparation and pharmaceutical compositions on which they are present Sanofi, Elf (FR) 1997-04-29 US disclosed
US-5340822-A Substance P, neurokinin antagonists ELF SANOFI (FR) 1994-08-23 US disclosed
EP-0512901-A1 Aminated polycyclic compounds and their enantiomers, process for their preparation and pharmaceutical compositions containing them SANOFI (FR) 1992-11-11 EP disclosed