SCHEMBL8296174

SCHEMBL8296174

COC(=O)c1c2cccc(-c3ccccc3O)c2nn1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
HPGD P15428 3/20 0.43
KDM4E B2RXH2 2/20 0.43
HSD17B10 Q99714 1/20 0.43
KDM4A O75164 1/20 0.42
CA12 O43570 2/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA9 Q16790 2/20 0.41
CA7 P43166 1/20 0.41
CA14 Q9ULX7 1/20 0.41
TOP2A P11388 1/20 0.41
PABPC1 P11940 1/20 0.40
EIF4H Q15056 1/20 0.40
TSHR P16473 2/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
IDO1 P14902 1/20 0.37
MAPT P10636 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3364448 0.82 BRD4 (0.47) ALDH1A1HPGDKDM4EHSD17B10PABPC1
SCHEMBL3364428 0.80 GABRG2 (0.41) ALDH1A1HPGDKDM4EHSD17B10CA12
SCHEMBL3367441 0.79 CRHR1 (0.47) ALDH1A1HPGDKDM4EHSD17B10LMNA
SCHEMBL3363110 0.79 KDM4E (0.41) ALDH1A1HPGDKDM4EHSD17B10LMNA
SCHEMBL3364893 0.79 SMN1; SMN2 (0.40) ALDH1A1HPGDKDM4EHSD17B10PABPC1
SCHEMBL3364882 0.79 ALDH1A1 (0.45) ALDH1A1HPGDKDM4EHSD17B10CA12
SCHEMBL3364407 0.79 HSD17B10 (0.44) ALDH1A1HPGDHSD17B10SMN1; SMN2MAPK14
SCHEMBL3364849 0.78 CRHR1 (0.43) KDM4ELMNASMN1; SMN2MAPTMEN1
SCHEMBL3362436 0.78 BRD9 (0.37) ALDH1A1HPGDKDM4EHSD17B10CA12
SCHEMBL3364215 0.78 GABRG2 (0.52) ALDH1A1HPGDKDM4EHSD17B10LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656353-B1 GABANERGIC MODULATORS HOFFMANN LA ROCHE (CH) 2010-01-27 EP disclosed
WO-2005016892-A1 GABANERGIC MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2005-02-24 WO disclosed