SCHEMBL8296292

SCHEMBL8296292

CS(=O)(=O)OCCC1(c2ccc(Cl)c(Cl)c2)CCC[N+]([O-])(Cc2ccccc2)C1

nearest known ligand 0.38

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 12/20 0.36
SLC6A3 Q01959 12/20 0.36
SLC6A2 P23975 6/20 0.36
TACR1 P25103 2/20 0.35
TACR2 P21452 1/20 0.35
TACR3 P29371 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8292836 0.85 TACR2 (0.34) SLC6A4SLC6A3SLC6A2TACR1TACR2
SCHEMBL8296079 0.76 CCR5 (0.52) TACR1TACR2TACR3
SCHEMBL8300821 0.73 SLC6A4 (0.37) SLC6A4SLC6A3SLC6A2TACR1TACR2
SCHEMBL8300818 0.73 CCR5 (0.43) SLC6A4SLC6A3SLC6A2TACR1
Hydrochloric Acid SCHEMBL8521991 0.73 CCR5 (0.42) SLC6A4SLC6A3SLC6A2TACR1
SCHEMBL6957564 0.72 TACR2 (0.54) TACR1TACR2TACR3
SCHEMBL6951866 0.72 TACR2 (0.62) TACR1TACR2TACR3
SCHEMBL8296291 0.72 TACR1 (0.63) TACR1TACR2TACR3
SCHEMBL8366952 0.70 TACR2 (0.47) TACR1TACR2TACR3
SCHEMBL8300346 0.70 TACR1 (0.45) TACR1TACR2TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0512901-B1 Aminated polycyclic compounds and their enantiomers, process for their preparation and pharmaceutical compositions containing them SANOFI SA (FR) 1999-06-23 EP disclosed
US-5770735-A Polycyclic amine compounds and their enantiomers, their method of preparation and pharmaceutical compositions in which they are present ELF SANOFI (FR) 1998-06-23 US disclosed
US-5625060-A Polycyclic amine compounds and their enantiomers, their method of preparation and pharmaceutical compositions on which they are present Sanofi, Elf (FR) 1997-04-29 US disclosed
US-5340822-A Substance P, neurokinin antagonists ELF SANOFI (FR) 1994-08-23 US disclosed
EP-0512901-A1 Aminated polycyclic compounds and their enantiomers, process for their preparation and pharmaceutical compositions containing them SANOFI (FR) 1992-11-11 EP disclosed