SCHEMBL8298554

SCHEMBL8298554

N#Cc1cc(Cl)c(C[N+](=O)[O-])cc1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 5/20 0.41
TRPV4 Q9HBA0 2/20 0.36
CYP1A2 P05177 1/20 0.33
MAPT P10636 1/20 0.33
ALOX15 P16050 1/20 0.33
GRIA1 P42261 1/20 0.33
GRIA2 P42262 1/20 0.33
GRIA3 P42263 1/20 0.33
GRIA4 P48058 1/20 0.33
DAO P14920 1/20 0.32
KHK P50053 1/20 0.32
IDH1 O75874 1/20 0.32
MRGPRX4 Q96LA9 1/20 0.31
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
KCNQ3 O43525 1/20 0.30
KCNQ2 O43526 1/20 0.30
KCNE1 P15382 1/20 0.30
KCNQ1 P51787 1/20 0.30
S1PR3 Q99500 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8298240 0.81 VCAM1 (0.44) VCAM1TRPV4CYP1A2MAPTALOX15
SCHEMBL23084780 0.78 TRPV4 (0.41) TRPV4DAOKHKIDH1MRGPRX4
SCHEMBL7744980 0.76 TDP1 (0.42) VCAM1MAPTALOX15ALDH1A1
SCHEMBL2725043 0.74 TRPV4 (0.38) TRPV4DAOKHKIDH1MRGPRX4
SCHEMBL297085 0.73 MRGPRX4 (0.41) TRPV4MRGPRX4KCNQ3KCNQ2KCNE1
SCHEMBL8299347 0.73 TRPV4 (0.41) VCAM1TRPV4CYP1A2MAPTALOX15
SCHEMBL1725293 0.72 VCAM1 (0.51) VCAM1TRPV4CYP1A2MAPTALOX15
SCHEMBL2731351 0.72 TRPV4 (0.39) TRPV4DAOKHKMRGPRX4CYP11B1
SCHEMBL8462168 0.71 TRPV4 (0.52) VCAM1TRPV4KHKCYP11B1CYP11B2
SCHEMBL8299664 0.71 TRPV4 (0.49) VCAM1TRPV4DAOCYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1227545-A 3-cyanoaryl pyrazoles and use thereof as herbicides BAYER AG (DE) 1999-09-01 CN disclosed
EP-0906285-A1 3-CYANOARYL PYRAZOLES AND USE THEREOF AS HERBICIDES BAYER AG (DE) 1999-04-07 EP disclosed
WO-1997046535-A1 3-CYANOARYL PYRAZOLES AND USE THEREOF AS HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 1997-12-11 WO disclosed