SCHEMBL8299347

SCHEMBL8299347

N#Cc1cc(F)c(CC[N+](=O)[O-])cc1F

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 2/20 0.41
VCAM1 P19320 3/20 0.33
ALDH1A1 P00352 1/20 0.33
GRIA1 P42261 2/20 0.30
GRIA2 P42262 2/20 0.30
GRIA3 P42263 2/20 0.30
GRIA4 P48058 2/20 0.30
CYP1A2 P05177 2/20 0.30
GRM6 O15303 1/20 0.30
MAPT P10636 1/20 0.30
ALOX15 P16050 1/20 0.30
XDH P47989 1/20 0.30
AKR1B1 P15121 1/20 0.30
DAO P14920 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17345635 0.81 ALDH1A1 (0.38) ALDH1A1CYP1A2MAPTCYP3A4CYP2C19
SCHEMBL5963451 0.74 ALDH1A1 (0.35) VCAM1ALDH1A1CYP1A2MAPTCYP3A4
SCHEMBL2731419 0.74 TRPV4 (0.47) TRPV4AKR1B1DAO
SCHEMBL13766377 0.73 TRPV4 (0.50) TRPV4AKR1B1DAO
SCHEMBL8298554 0.73 VCAM1 (0.41) TRPV4VCAM1ALDH1A1GRIA1GRIA2
SCHEMBL4614436 0.70 VCAM1 (0.47) TRPV4VCAM1ALDH1A1GRIA1GRIA2
SCHEMBL8298240 0.70 VCAM1 (0.44) TRPV4VCAM1ALDH1A1GRIA1GRIA2
SCHEMBL365265 0.70 TRPV4 (0.50) TRPV4AKR1B1
SCHEMBL3161291 0.70 TRPV4 (0.50) TRPV4
SCHEMBL363766 0.70 TRPV4 (0.50) TRPV4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0906285-A1 3-CYANOARYL PYRAZOLES AND USE THEREOF AS HERBICIDES BAYER AG (DE) 1999-04-07 EP disclosed
EP-0897383-A1 3-CYANOARYL PYRAZOLES AND THEIR USE AS HERBICIDES BAYER AG (DE) 1999-02-24 EP disclosed
WO-1997046535-A1 3-CYANOARYL PYRAZOLES AND USE THEREOF AS HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 1997-12-11 WO disclosed
WO-1997040018-A1 3-CYANOARYL PYRAZOLES AND THEIR USE AS HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 1997-10-30 WO disclosed